SCHEMBL740864

SCHEMBL740864

CON(C)C(=O)[C@@H](Cc1ccc(Br)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 7/20 0.60
CTSK P43235 6/20 0.60
JAK3 P52333 1/20 0.51
BTK Q06187 1/20 0.51
CTSB P07858 2/20 0.46
CTSL P07711 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
CACNA1B Q00975 1/20 0.46
ITGB3 P05106 1/20 0.45
ITGA2B P08514 1/20 0.45
ACE P12821 1/20 0.45
AAK1 Q2M2I8 2/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
FAAH O00519 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740863 1.00 CTSS (0.60) CTSSCTSKJAK3BTKCTSB
SCHEMBL13977456 1.00 CTSS (0.60) CTSSCTSKJAK3BTKCTSB
SCHEMBL9963893 0.89 CTSS (0.60) CTSSCTSKJAK3BTKCTSB
SCHEMBL7033260 0.88 PPARG (0.52) CTSSCTSKJAK3BTKCTSB
SCHEMBL3878792 0.88 CTSS (0.60) CTSSCTSKJAK3BTKCTSB
SCHEMBL6345086 0.88 JAK3 (0.51) CTSSCTSKJAK3BTKCTSB
SCHEMBL268923 0.88 JAK3 (0.51) CTSSCTSKJAK3BTKCTSB
SCHEMBL7033261 0.88 PPARG (0.52) CTSSCTSKJAK3BTKCTSB
SCHEMBL3989315 0.88 CTSS (0.60) CTSSCTSKJAK3BTKCTSB
SCHEMBL6557659 0.88 JAK3 (0.61) CTSSCTSKJAK3BTKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed