SCHEMBL7408809

SCHEMBL7408809

OCc1ccc(CCN2CCC2)cn1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 10/20 0.59
CYP1A2 P05177 2/20 0.57
CYP2D6 P10635 1/20 0.57
L3MBTL1 Q9Y468 2/20 0.46
MBTD1 Q05BQ5 1/20 0.46
L3MBTL3 Q96JM7 1/20 0.46
TDP1 Q9NUW8 1/20 0.45
CYP3A4 P08684 1/20 0.44
SLC6A3 Q01959 1/20 0.43
SIGMAR1 Q99720 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13569223 0.84 HRH3 (0.72) HRH3CYP1A2CYP2D6L3MBTL1MBTD1
SCHEMBL23530205 0.83 HRH3 (0.47) HRH3CYP1A2CYP2D6L3MBTL1MBTD1
SCHEMBL2886050 0.83 CYP1A2 (0.73) HRH3CYP1A2CYP2D6L3MBTL1MBTD1
SCHEMBL21414430 0.77 HRH3 (0.58) HRH3CYP1A2CYP2D6SIGMAR1
SCHEMBL7399231 0.77 HRH3 (0.50) HRH3CYP1A2CYP2D6L3MBTL1MBTD1
SCHEMBL23530102 0.75 LTA4H (0.63) HRH3
SCHEMBL12668355 0.74 CYP1A2 (0.75) HRH3CYP1A2CYP2D6L3MBTL1MBTD1
SCHEMBL6921327 0.74 HRH3 (0.72) HRH3CYP1A2CYP2D6L3MBTL1MBTD1
SCHEMBL13990825 0.74 HRH3 (1.00) HRH3CYP1A2CYP2D6L3MBTL1MBTD1
SCHEMBL4625412 0.73 HRH3 (0.54) HRH3CYP1A2CYP2D6L3MBTL1MBTD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002042305-A1 NITROGEN SUBSTITUTED 1,2,4-TRIAZOLO[3,4-A]PHTHALAZINE DERIVATIVES FOR ENHANCING COGNITION MERCK SHARP & DOHME LIMITED (GB) 2002-05-30 WO disclosed