SCHEMBL7399231

SCHEMBL7399231

Brc1ccc(CCN2CCC2)cn1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 8/20 0.50
CYP1A2 P05177 2/20 0.49
CYP2D6 P10635 1/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
MBTD1 Q05BQ5 1/20 0.49
L3MBTL3 Q96JM7 1/20 0.49
TDP1 Q9NUW8 1/20 0.47
CYP3A4 P08684 1/20 0.46
SLC6A3 Q01959 2/20 0.46
SIGMAR1 Q99720 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4625412 0.97 HRH3 (0.54) HRH3CYP1A2CYP2D6L3MBTL1MBTD1
SCHEMBL227159 0.95 HRH3 (0.56) HRH3CYP1A2CYP2D6L3MBTL1MBTD1
SCHEMBL2930854 0.85 CHRNB2 (0.51) HRH3CYP1A2CYP2D6TDP1CYP3A4
SCHEMBL2532973 0.85 SIGMAR1 (0.53) HRH3L3MBTL3SIGMAR1
SCHEMBL29725200 0.79 HRH3 (0.55) HRH3CYP2D6L3MBTL1MBTD1L3MBTL3
SCHEMBL3869875 0.79 HRH3 (0.55) HRH3CYP2D6L3MBTL1MBTD1L3MBTL3
SCHEMBL1858355 0.77 HRH3 (0.59) HRH3CYP2D6TDP1
SCHEMBL31093419 0.77 HRH3 (0.59) HRH3CYP2D6TDP1
SCHEMBL7408809 0.77 HRH3 (0.59) HRH3CYP1A2CYP2D6L3MBTL1MBTD1
SCHEMBL8281118 0.76 HRH3 (0.61) HRH3CYP1A2CYP2D6L3MBTL1MBTD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002042305-A1 NITROGEN SUBSTITUTED 1,2,4-TRIAZOLO[3,4-A]PHTHALAZINE DERIVATIVES FOR ENHANCING COGNITION MERCK SHARP & DOHME LIMITED (GB) 2002-05-30 WO disclosed