SCHEMBL7409096

SCHEMBL7409096

CC(C)(C)OC(=O)CC(NC(=O)C1(C(=O)NC(CCC(=O)O)C(=O)Nc2cccc(Oc3ccccc3)c2)CCC1)C(O)COc1c(F)c(F)cc(F)c1F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 5/20 0.35
HDAC4 P56524 3/20 0.33
HDAC1 Q13547 2/20 0.33
SIRT5 Q9NXA8 1/20 0.33
CASP3 P42574 2/20 0.33
CASP6 P55212 1/20 0.33
CASP8 Q14790 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC9 Q9UKV0 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33
MMP2 P08253 1/20 0.33
MMP3 P08254 1/20 0.33
MMP10 P09238 1/20 0.33
MMP9 P14780 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7404576 0.94 KDR (0.34) KDRHDAC4HDAC1CASP3CASP6
SCHEMBL7410069 0.93 HDAC4 (0.33) KDRHDAC4HDAC1CASP3CASP6
SCHEMBL7405678 0.93 KDR (0.35) KDRHDAC4HDAC1HDAC3HDAC7
SCHEMBL7409725 0.89 CASP3 (0.43) CASP3CASP6CASP8
SCHEMBL7404413 0.83 CASP3 (0.40) CASP3CASP6CASP8
SCHEMBL7402840 0.82 CASP3 (0.41) CASP3CASP6CASP8
SCHEMBL7451783 0.82 CASP3 (0.39) KDRCASP3CASP6CASP8MMP8
SCHEMBL7403799 0.82 CASP3 (0.49) CASP3CASP6CASP8
SCHEMBL7404112 0.80 CASP3 (0.48) CASP3CASP6CASP8
SCHEMBL7405838 0.79 HPGD (0.37) HDAC4HDAC1CASP3CASP6CASP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002076968-A1 MALONATES AS INHIBITORS OF THE ICE/CED-6 FAMILY OF CYSTEINE PROTEASES NOVARTIS AG (CH) 2002-10-03 WO disclosed