SCHEMBL7409173

SCHEMBL7409173

CCC(C(=O)O)N1CCN(S(=O)(=O)Cc2ccccc2)CC1=O

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.50
GAA P10253 1/20 0.50
CYP2C19 P33261 1/20 0.50
GCK P35557 1/20 0.50
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 1/20 0.47
KMT2A Q03164 1/20 0.47
RAB9A P51151 1/20 0.46
HPGD P15428 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
PKM P14618 2/20 0.45
HSD11B1 P28845 1/20 0.44
MAPT P10636 1/20 0.44
HSD17B10 Q99714 1/20 0.44
MAPK1 P28482 1/20 0.43
LMNA P02545 1/20 0.43
RORC P51449 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7397071 0.89 TSHR (0.52) TSHRGAACYP2C19ALDH1A1KDM4E
SCHEMBL7365043 0.74 KMT2A (0.52) TSHRGAACYP2C19ALDH1A1KDM4E
SCHEMBL735675 0.71 TSHR (0.81) TSHRGAACYP2C19ALDH1A1KMT2A
SCHEMBL18711922 0.68 TSHR (0.70) TSHRGAACYP2C19ALDH1A1KDM4E
N-Benzylmethylamine SCHEMBL29834172 0.68 LMNA (0.53) ALDH1A1KDM4EKMT2APKMMAPT
SCHEMBL10077130 0.67 L3MBTL1 (0.71) TSHRGAACYP2C19ALDH1A1KDM4E
SCHEMBL12067603 0.67 TSHR (0.63) TSHRGAACYP2C19ALDH1A1KDM4E
SCHEMBL18702279 0.65 TSHR (0.65) TSHRGAACYP2C19ALDH1A1KDM4E
SCHEMBL6738518 0.65 TSHR (0.96) TSHRGAACYP2C19ALDH1A1KDM4E
SCHEMBL12384638 0.65 NPSR1 (0.60) TSHRGAACYP2C19ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211183-B1 PIPERAZINE DERIVATIVE ANTICOAGULANTS; ANTIISCHEMIC AGENTS; CARDIOVASCULAR DISORDERS COR THERAPEUTICS, INC. 2001-04-03 US disclosed
EP-0975625-A1 SELECTIVE FACTOR Xa INHIBITORS COR THERAPEUTICS, INC. (US) 2000-02-02 EP disclosed
WO-1998046591-A1 SELECTIVE FACTOR Xa INHIBITORS COR THERAPEUTICS, INC. (US) 1998-10-22 WO disclosed