SCHEMBL7409889

SCHEMBL7409889

CC(C)c1ccc2[nH]c(C3CCCN3)nc2c1OC(=O)O

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 0.50
SCN10A Q9Y5Y9 1/20 0.39
CDC7 O00311 4/20 0.37
PIM1 P11309 4/20 0.37
CSNK2B P67870 4/20 0.37
CSNK2A1 P68400 4/20 0.37
PARP2 Q9UGN5 1/20 0.35
CIT O14578 1/20 0.35
CYP1A2 P05177 1/20 0.35
CSNK2A2 P19784 1/20 0.35
GSK3B P49841 1/20 0.35
DYRK1A Q13627 1/20 0.35
CSNK2A3 Q8NEV1 1/20 0.35
TAOK3 Q9H2K8 1/20 0.35
ERCC1 P07992 1/20 0.34
ERCC4 Q92889 1/20 0.34
PTGES O14684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7415905 0.81 PARP1 (0.50) PARP1PARP2
SCHEMBL7415820 0.75 PARP1 (0.56) PARP1SCN10ACDC7PIM1CSNK2B
SCHEMBL6869338 0.69 PARP1 (0.69) PARP1PIM1PARP2DYRK1A
SCHEMBL7702651 0.67 PARP1 (1.00) PARP1PARP2
SCHEMBL630259 0.67 PARP1 (1.00) PARP1PARP2
SCHEMBL633643 0.67 PARP1 (1.00) PARP1PARP2
SCHEMBL1298158 0.67 PARP1 (0.80) PARP1PIM1PARP2DYRK1A
SCHEMBL15844095 0.67 PARP1 (0.53) PARP1SCN10ACDC7PIM1CSNK2B
SCHEMBL15844096 0.67 PARP1 (0.53) PARP1SCN10ACDC7PIM1CSNK2B
SCHEMBL18596118 0.66 SCN10A (0.55) PARP1SCN10ACDC7PIM1CSNK2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed