SCHEMBL7415905

SCHEMBL7415905

CC(C)c1ccc2[nH]c(C3CCNC3)nc2c1OC(=O)O

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 16/20 0.50
PARP2 Q9UGN5 2/20 0.38
TLR9 Q9NR96 2/20 0.34
TLR8 Q9NR97 2/20 0.34
TLR7 Q9NYK1 2/20 0.34
HTR1F P30939 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7409889 0.81 PARP1 (0.50) PARP1PARP2
SCHEMBL7408785 0.76 PARP1 (0.57) PARP1PARP2
SCHEMBL7411360 0.75 PARP1 (0.56) PARP1PARP2
SCHEMBL7413860 0.70 PARP1 (0.60) PARP1PARP2TLR9TLR8TLR7
SCHEMBL7421139 0.69 PARP1 (0.60) PARP1PARP2
SCHEMBL7416833 0.69 PARP1 (0.57) PARP1PARP2
SCHEMBL6869625 0.69 PARP1 (0.69) PARP1PARP2
SCHEMBL7410253 0.68 PARP1 (0.57) PARP1PARP2
SCHEMBL631186 0.67 PARP1 (1.00) PARP1PARP2
SCHEMBL7045124 0.64 PARP1 (0.53) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed