SCHEMBL741000

SCHEMBL741000

COCCCn1c([C@@H]2CCCNC2)nc2cc(Cl)c(Cl)cc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 2/20 0.49
HRH1 P35367 2/20 0.49
PRPS1 P60891 1/20 0.42
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
BRD4 O60885 2/20 0.39
REN P00797 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
SOS1 Q07889 1/20 0.37
KCNH2 Q12809 1/20 0.37
CCNT1 O60563 1/20 0.36
CDK7 P50613 1/20 0.36
CDK9 P50750 1/20 0.36
CCNH P51946 1/20 0.36
MNAT1 P51948 1/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
JAK3 P52333 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741001 1.00 CHRM1 (0.49) CHRM1HRH1PRPS1HTR2AHTR2C
SCHEMBL740755 0.88 HRH1 (0.52) CHRM1HRH1BRD4RENKCNH2
SCHEMBL740756 0.88 HRH1 (0.52) CHRM1HRH1BRD4RENKCNH2
SCHEMBL741972 0.84 HRH1 (0.53) CHRM1HRH1BRD4RENJAK2
SCHEMBL741971 0.84 HRH1 (0.53) CHRM1HRH1BRD4RENJAK2
SCHEMBL737976 0.84 HRH1 (0.55) CHRM1HRH1BRD4RENKCNH2
SCHEMBL742774 0.84 HRH1 (0.54) CHRM1HRH1BRD4RENKCNH2
SCHEMBL740741 0.84 HRH1 (0.54) CHRM1HRH1PRPS1BRD4REN
SCHEMBL742773 0.84 HRH1 (0.54) CHRM1HRH1BRD4RENKCNH2
SCHEMBL737977 0.84 HRH1 (0.55) CHRM1HRH1BRD4RENKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed