SCHEMBL741972

SCHEMBL741972

COCCCn1c(C2CCCNC2)nc2cc(C)ccc21

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 3/20 0.53
CHRM1 P11229 2/20 0.53
P2RX3 P56373 1/20 0.43
REN P00797 3/20 0.42
JAK2 O60674 5/20 0.41
JAK1 P23458 5/20 0.41
TYK2 P29597 5/20 0.41
JAK3 P52333 5/20 0.41
BRD4 O60885 2/20 0.40
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
TLR8 Q9NR97 1/20 0.38
OPRM1 P35372 2/20 0.37
OPRD1 P41143 2/20 0.37
OPRK1 P41145 2/20 0.37
OPRL1 P41146 2/20 0.37
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741971 1.00 HRH1 (0.53) HRH1CHRM1P2RX3RENJAK2
SCHEMBL740741 0.89 HRH1 (0.54) HRH1CHRM1P2RX3RENJAK2
SCHEMBL740742 0.89 HRH1 (0.54) HRH1CHRM1P2RX3RENJAK2
SCHEMBL762533 0.89 CHRM1 (0.51) HRH1CHRM1P2RX3JAK2JAK1
SCHEMBL739842 0.86 HRH1 (0.70) HRH1CHRM1RENBRD4OPRM1
SCHEMBL739843 0.86 HRH1 (0.70) HRH1CHRM1RENBRD4OPRM1
SCHEMBL741000 0.84 CHRM1 (0.49) HRH1CHRM1RENJAK2JAK1
SCHEMBL741001 0.84 CHRM1 (0.49) HRH1CHRM1RENJAK2JAK1
Piperidine SCHEMBL742276 0.84 HRH1 (0.67) HRH1CHRM1RENOPRM1OPRD1
SCHEMBL740756 0.83 HRH1 (0.52) HRH1CHRM1RENBRD4OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed