SCHEMBL7410024

SCHEMBL7410024

CCOC(=O)Nc1ccc(OC)cc1C(C)=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
ALDH1A1 P00352 7/20 0.55
HPGD P15428 4/20 0.54
HSD17B10 Q99714 3/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
MTNR1B P49286 2/20 0.53
KMT2A Q03164 3/20 0.50
MAPK1 P28482 2/20 0.50
MEN1 O00255 2/20 0.50
CYP3A4 P08684 1/20 0.50
NPC1 O15118 1/20 0.49
HTT P42858 1/20 0.49
LMNA P02545 1/20 0.48
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
TSHR P16473 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
ALOX15 P16050 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4481689 0.83 ALDH1A1 (0.57) ALDH1A1HPGDSMN1; SMN2KMT2AMAPK1
SCHEMBL2090279 0.82 CYP1A2 (0.58) CYP1A2CYP2C9CYP2C19ALDH1A1HSD17B10
SCHEMBL1026559 0.82 ALDH1A1 (0.59) ALDH1A1HPGDSMN1; SMN2MTNR1BKMT2A
SCHEMBL12575809 0.81 CYP1A2 (0.56) CYP1A2CYP2C9CYP2C19ALDH1A1HPGD
SCHEMBL7557552 0.81 CYP1A2 (0.56) CYP1A2CYP2C9CYP2C19ALDH1A1HPGD
SCHEMBL10489963 0.80 AKR1C3 (0.57) CYP1A2CYP2C9CYP2C19ALDH1A1SMN1; SMN2
SCHEMBL7254155 0.79 ALDH1A1 (0.54) CYP1A2CYP2C9CYP2C19ALDH1A1HPGD
SCHEMBL7413878 0.79 ALDH1A1 (0.60) CYP1A2CYP2C9CYP2C19ALDH1A1HPGD
SCHEMBL18024095 0.79 ALDH1A1 (0.54) CYP1A2CYP2C9CYP2C19ALDH1A1HPGD
SCHEMBL29648996 0.78 NLRP3 (0.54) CYP1A2CYP2C9CYP2C19ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0107398-B1 ORTHO SUBSTITUTED DIHYDROXY-2(1H)QUINAZOLINONE-1-ALKANOIC ACIDS ORTHO PHARMA CORP (US) 1988-06-08 EP disclosed
US-4631283-A RENAL VASODILATORS, CARDIOVASCULAR AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1986-12-23 US disclosed
US-4490374-A CARDIOVASCULAR AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1984-12-25 US disclosed
EP-0107398-A1 Ortho substituted dihydroxy-2(1H)quinazolinone-1-alkanoic acids ORTHO PHARMACEUTICAL CORPORATION (US) 1984-05-02 EP disclosed