SCHEMBL7410146

SCHEMBL7410146

CCCN1CCC(c2nc3c(C)c(CC)ccc3[nH]2)CC1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 11/20 0.61
PARP2 Q9UGN5 1/20 0.60
TLR9 Q9NR96 2/20 0.44
TLR8 Q9NR97 2/20 0.44
TLR7 Q9NYK1 2/20 0.44
DRD2 P14416 4/20 0.41
HTR1F P30939 1/20 0.39
SLC6A4 P31645 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7409701 0.94 PARP1 (0.61) PARP1PARP2TLR9TLR8TLR7
SCHEMBL7410700 0.87 PARP1 (0.57) PARP1PARP2DRD2
SCHEMBL7409815 0.82 PARP1 (0.60) PARP1PARP2TLR9TLR8TLR7
SCHEMBL7409390 0.79 PARP1 (0.58) PARP1PARP2DRD2
SCHEMBL7415524 0.78 TSHR (0.39) PARP1PARP2DRD2
SCHEMBL423949 0.75 PARP1 (1.00) PARP1PARP2
SCHEMBL7409877 0.73 PARP1 (0.55) PARP1PARP2HTR1F
SCHEMBL6865071 0.73 PARP1 (0.73) PARP1PARP2
SCHEMBL7413860 0.72 PARP1 (0.60) PARP1PARP2TLR9TLR8TLR7
Succinic Acid SCHEMBL29396818 0.71 PARP1 (0.90) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed