Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | MAPT | P10636 | 7/20 | 0.39 |
| ▸ | CACNA1C | Q13936 | 5/20 | 0.39 |
| ▸ | CYP1A2 | P05177 | 4/20 | 0.39 |
| ▸ | CYP3A4 | P08684 | 4/20 | 0.39 |
| ▸ | ADORA3 | P0DMS8 | 4/20 | 0.39 |
| ▸ | CYP2C9 | P11712 | 4/20 | 0.39 |
| ▸ | CYP2C19 | P33261 | 4/20 | 0.39 |
| ▸ | KMT2A | Q03164 | 4/20 | 0.39 |
| ▸ | TSHR | P16473 | 3/20 | 0.39 |
| ▸ | NFKB1 | P19838 | 3/20 | 0.39 |
| ▸ | CYP2D6 | P10635 | 2/20 | 0.39 |
| ▸ | MEN1 | O00255 | 2/20 | 0.39 |
| ▸ | BACE1 | P56817 | 3/20 | 0.35 |
| ▸ | CYP2A6 | P11509 | 1/20 | 0.35 |
| ▸ | CACNA1B | Q00975 | 5/20 | 0.35 |
| ▸ | ALDH1A1 | P00352 | 2/20 | 0.33 |
| ▸ | HPGD | P15428 | 2/20 | 0.33 |
| ▸ | TDP1 | Q9NUW8 | 2/20 | 0.33 |
| ▸ | KDM4E | B2RXH2 | 1/20 | 0.33 |
| ▸ | ABCC4 | O15439 | 1/20 | 0.33 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL7409728 | 1.00 | MAPT (0.39) | MAPTCACNA1CCYP1A2CYP3A4ADORA3 | |
| SCHEMBL7407834 | 1.00 | MAPT (0.39) | MAPTCACNA1CCYP1A2CYP3A4ADORA3 | |
| SCHEMBL10372051 | 0.88 | CYP2A6 (0.42) | MAPTCACNA1CKMT2AMEN1BACE1 | |
| SCHEMBL29389135 | 0.86 | MAPT (0.54) | MAPTCACNA1CCYP1A2CYP3A4ADORA3 | |
| SCHEMBL29389617 | 0.84 | CACNA1C (0.42) | MAPTCACNA1CCYP1A2CYP3A4ADORA3 | |
| SCHEMBL29388969 | 0.84 | MAPT (0.46) | MAPTCACNA1CCYP1A2CYP3A4ADORA3 | |
| SCHEMBL29390127 | 0.84 | MAPT (0.46) | MAPTCACNA1CCYP1A2CYP3A4ADORA3 | |
| SCHEMBL29389652 | 0.84 | MAPT (0.46) | MAPTCACNA1CCYP1A2CYP3A4ADORA3 | |
| SCHEMBL29386583 | 0.83 | CACNA1C (0.44) | MAPTCACNA1CCYP1A2CYP3A4ADORA3 | |
| SCHEMBL29819617 | 0.83 | CACNA1C (0.41) | MAPTCACNA1CCYP1A2CYP3A4ADORA3 |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| US-20140088056-A1 | CARDIAC GLYCOSIDES ARE POTENT INHIBITORS OF INTERFERON-BETA GENE EXPRESSION | PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) | 2014-03-27 | — | — | US | claimed |
| WO-2012050884-A2 | CARDIAC GLYCOSIDES ARE POTENT INHIBITORS OF INTERFERON-BETA GENE EXPRESSION | PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) | 2012-04-19 | — | — | WO | claimed |
| US-11963964-B2 | Small molecules for mouse satellite cell proliferation | PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) | 2024-04-23 | — | — | US | disclosed |
| US-20220054499-A1 | SMALL MOLECULES FOR MOUSE SATELLITE CELL PROLIFERATION | PRESIDENT AND FELLOWS OF HARVARD COLLEGE | 2022-02-24 | — | — | US | disclosed |
| US-11026952-B2 | Small molecules for mouse satellite cell proliferation | PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) | 2021-06-08 | — | — | US | disclosed |
| US-20200352957-A1 | SMALL MOLECULE SCREENING FOR MOUSE SATELLITE CELL PROLIFERATION | PRESIDENT AND FELLOWS OF HARVARD COLLEGE | 2020-11-12 | — | — | US | disclosed |
| US-10660902-B2 | Method of increasing satellite cell proliferation with an HDAC inhibitor | PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) | 2020-05-26 | — | — | US | disclosed |
| EP-3411040-A1 | SMALL MOLECULES FOR MOUSE SATELLITE CELL PROLIFERATION | President and Fellows of Harvard College (US) | 2018-12-12 | — | — | EP | disclosed |
| US-20180153902-A1 | SMALL MOLECULE SCREENING FOR MOUSE SATELLITE CELL PROLIFERATION | HOWARD HUGHES MEDICAL INSTITUTE | 2018-06-07 | — | — | US | disclosed |
| US-9782417-B2 | Methods of increasing satellite cell proliferation with kinase inhibitors | PRESIDENTS AND FELLOWS OF HARVARD COLLEGE (US) | 2017-10-10 | — | — | US | disclosed |
| WO-2017136480-A1 | SMALL MOLECULES FOR MOUSE SATELLITE CELL PROLIFERATION | PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) | 2017-08-10 | — | — | WO | disclosed |
| US-9248185-B2 | Methods of increasing satellite cell proliferation | PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) | 2016-02-02 | — | — | US | disclosed |
| US-20140294855-A1 | SMALL MOLECULE SCREENING FOR MOUSE SATELLITE CELL PROLIFERATION | PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) | 2014-10-02 | — | — | US | disclosed |
| US-20140088056-A1 | CARDIAC GLYCOSIDES ARE POTENT INHIBITORS OF INTERFERON-BETA GENE EXPRESSION | PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) | 2014-03-27 | — | — | US | disclosed |
| EP-2646107-A2 | AGENT DELIVERY SYSTEMS FOR SELECTIVE NEUROMODULATION | Spinal Modulation Inc. (US) | 2013-10-09 | — | — | EP | disclosed |
| WO-2012174537-A2 | SMALL MOLECULE SCREENING FOR MOUSE SATELLITE CELL PROLIFERATION | PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) | 2012-12-20 | — | — | WO | disclosed |
| US-20120310140-A1 | DIRECTED DELIVERY OF AGENTS TO NEURAL ANATOMY | SPINAL MODULATION, INC. (US) | 2012-12-06 | — | — | US | disclosed |
| WO-2012075337-A2 | DIRECTED DELIVERY OF AGENTS TO NEURAL ANATOMY | SPINAL MODULATION, INC. (US) | 2012-06-07 | — | — | WO | disclosed |
| WO-2012050884-A2 | CARDIAC GLYCOSIDES ARE POTENT INHIBITORS OF INTERFERON-BETA GENE EXPRESSION | PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) | 2012-04-19 | — | — | WO | disclosed |
| US-4902694-A | TREATING CONGESTIVE HEART FAILURE | ELI LILLY AND COMPANY (US) | 1990-02-20 | — | — | US | disclosed |
Patent text — is the patent's own abstract consistent with the prediction?
For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.
| Patent | Title | Text reads most about | Predicted target · text-rank |
|---|---|---|---|
| US-11026952-B2 | Small molecules for mouse satellite cell proliferation | MKI67, MYLK2, MYH2 | MAPT 4150/4885CACNA1C 2996/4885CYP1A2 4849/4885 |
| US-10660902-B2 | Method of increasing satellite cell proliferation with an HDAC inhibitor | HDAC4, HDAC1, HDAC5 | MAPT 3910/4885CACNA1C 3447/4885CYP1A2 4694/4885 |
| US-20220054499-A1 | SMALL MOLECULES FOR MOUSE SATELLITE CELL PROLIFERATION | MKI67, MYLK2, MYH2 | MAPT 4150/4885CACNA1C 2996/4885CYP1A2 4849/4885 |
| US-20180153902-A1 | SMALL MOLECULE SCREENING FOR MOUSE SATELLITE CELL PROLIFERATION | MKI67, MYLK2, MYH2 | MAPT 4009/4885CACNA1C 2730/4885CYP1A2 4811/4885 |
| US-11963964-B2 | Small molecules for mouse satellite cell proliferation | MKI67, MYLK2, MYH2 | MAPT 4150/4885CACNA1C 2996/4885CYP1A2 4849/4885 |
| US-20200352957-A1 | SMALL MOLECULE SCREENING FOR MOUSE SATELLITE CELL PROLIFERATION | MKI67, MYLK2, MYH2 | MAPT 4009/4885CACNA1C 2730/4885CYP1A2 4811/4885 |
| US-20140294855-A1 | SMALL MOLECULE SCREENING FOR MOUSE SATELLITE CELL PROLIFERATION | MKI67, MYLK2, MYH2 | MAPT 3922/4885CACNA1C 2559/4885CYP1A2 4795/4885 |
| US-20140088056-A1 | CARDIAC GLYCOSIDES ARE POTENT INHIBITORS OF INTERFERON-BETA GENE EXPRESSION | IRF3, IFNG, STING1 | MAPT 4814/4885CACNA1C 154/4885CYP1A2 2870/4885 |
“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.