SCHEMBL7411328

SCHEMBL7411328

O=C(O)CC(NC(=O)C1(C(=O)NC(CCC(=O)OCc2ccccc2)C(=O)Nc2cccc(Oc3ccccc3)c2)CCC1)C(=O)COc1c(F)c(F)cc(F)c1F

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 20/20 0.44
CASP8 Q14790 17/20 0.44
CASP6 P55212 14/20 0.44
CASP1 P29466 3/20 0.42
CASP9 P55211 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7406778 0.93 CASP3 (0.47) CASP3CASP8CASP6
SCHEMBL7451783 0.93 CASP3 (0.39) CASP3CASP8CASP6
SCHEMBL7404112 0.92 CASP3 (0.48) CASP3CASP8CASP6
SCHEMBL7403799 0.92 CASP3 (0.49) CASP3CASP8CASP6CASP1CASP9
SCHEMBL7406976 0.91 CASP3 (0.45) CASP3CASP8CASP6
SCHEMBL7404243 0.91 CASP3 (0.46) CASP3CASP8CASP6CASP1CASP9
SCHEMBL7402816 0.91 CASP3 (0.48) CASP3CASP8CASP6CASP1CASP9
SCHEMBL7463728 0.90 CASP3 (0.50) CASP3CASP8CASP6CASP1CASP9
SCHEMBL7454999 0.90 CASP3 (0.48) CASP3CASP8CASP6CASP1CASP9
SCHEMBL7408942 0.89 CASP3 (0.49) CASP3CASP8CASP6CASP1CASP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002076968-A1 MALONATES AS INHIBITORS OF THE ICE/CED-6 FAMILY OF CYSTEINE PROTEASES NOVARTIS AG (CH) 2002-10-03 WO disclosed