SCHEMBL7411485

SCHEMBL7411485

Cc1cc(NC(=O)N2CCc3cc4c(cc32)CCN4C)c2ccccc2n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
MAPT P10636 1/20 0.53
NFKB1 P19838 1/20 0.53
BLM P54132 1/20 0.53
PMP22 Q01453 1/20 0.53
USP2 O75604 1/20 0.52
LMNA P02545 2/20 0.51
NPSR1 Q6W5P4 1/20 0.51
HTT P42858 3/20 0.50
HTR2C P28335 3/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.47
GALR3 O60755 1/20 0.47
RAB9A P51151 1/20 0.47
IGF1R P08069 1/20 0.46
HTR1A P08908 1/20 0.44
HTR1D P28221 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8526774 0.86 HTR2B (0.72) HTR2BCYP1A2CYP3A4MAPTNFKB1
SCHEMBL7420874 0.85 MAPT (0.59) HTR2BCYP1A2CYP3A4MAPTNFKB1
SCHEMBL9049984 0.83 MAPT (0.49) HTR2BCYP1A2CYP3A4MAPTNFKB1
SCHEMBL8529863 0.83 HTR2C (0.56) HTR2BCYP1A2CYP3A4MAPTNFKB1
SCHEMBL7474827 0.77 HTR2C (0.58) HTR2BCYP1A2CYP3A4MAPTNFKB1
SCHEMBL9051003 0.75 HTT (0.46) HTR2BCYP1A2CYP3A4MAPTNFKB1
SCHEMBL29462322 0.72 HTR2B (0.87) HTR2BCYP1A2CYP3A4MAPTNFKB1
SCHEMBL4855474 0.71 HTT (0.75) MAPTHTTMEN1KMT2ASMN1; SMN2
SCHEMBL7423705 0.70 HTR2C (0.76) HTR2BCYP1A2CYP3A4MAPTBLM
SCHEMBL5053541 0.70 HTT (0.73) CYP1A2MAPTHTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994004533-A1 CONDENSED INDOLE DERIVATIVES AS 5HT2C AND 5HT2B ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-03-03 WO disclosed