SCHEMBL7412280

SCHEMBL7412280

CC(=O)C(=CN(C)C)c1cnc2c(c1)CN(C)C(=O)N2C

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FGFR4 P22455 2/20 0.34
HPGD P15428 2/20 0.33
GFER P55789 1/20 0.33
FGFR1 P11362 1/20 0.32
ALDH1A1 P00352 2/20 0.32
HTT P42858 1/20 0.32
KDM4E B2RXH2 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7415711 0.78 BRD4 (0.32)
SCHEMBL7328560 0.74 GABRG2 (0.36)
SCHEMBL7419734 0.71 ENPP1 (0.31)
SCHEMBL7413265 0.70 HSD17B10 (0.46) HPGDALDH1A1HTTKDM4E
SCHEMBL7421949 0.69 BRD4 (0.40) FGFR4FGFR1
SCHEMBL7442306 0.68 BRD4 (0.50) HPGDGFERALDH1A1HTT
SCHEMBL7315582 0.68 ALDH1A1 (0.36) HPGDALDH1A1
SCHEMBL7473009 0.67 XIAP (0.45)
SCHEMBL7835908 0.62 RECQL (0.48) HPGDALDH1A1HTTKDM4EMAPT
SCHEMBL22440125 0.62 RECQL (0.48) HPGDALDH1A1HTTKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5002944-A Compounds having cardiotonic activity RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-03-26 US disclosed
EP-0333727-A1 HETEROCYCLIC SUBSTITUTED BICYCLOUREAS HAVING CARDIOTONIC ACTIVITY RORER INTERNATIONAL (OVERSEAS) INC. (a Delaware corporation) (US) 1989-09-27 EP disclosed
US-4859672-A Pyrido[2,3-d]pyrimidinone and imidazo[4,5-b]pyrimidinone RORER PHARMACEUTICAL CORPORATION (US) 1989-08-22 US disclosed
WO-1988003025-A1 HETEROCYCLIC SUBSTITUTED BICYCLOUREAS HAVING CARDIOTONIC ACTIVITY RORER INTERNATIONAL (OVERSEAS) INC. (US) 1988-05-05 WO disclosed