SCHEMBL7412563

SCHEMBL7412563

COc1cc(C)c(S(=O)(=O)N[C@@H](Cc2ccc(OCCCONC(=N)N)cc2)C(=O)O)c(C)c1C

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AVPR1B P47901 7/20 0.51
AVPR1A P37288 9/20 0.49
PLG P00747 1/20 0.48
ITGB3 P05106 1/20 0.46
ITGA2B P08514 1/20 0.46
F2 P00734 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL7412254 0.96 AVPR1B (0.48) AVPR1BAVPR1APLGITGB3ITGA2B
SCHEMBL7414099 0.88 ITGB3 (0.53) ITGB3ITGA2B
SCHEMBL7418575 0.88 ITGB3 (0.55) ITGB3ITGA2B
SCHEMBL7412260 0.88 AVPR1A (0.45) AVPR1BAVPR1APLG
SCHEMBL7463784 0.84 ITGB3 (0.48) ITGB3ITGA2B
Trifluoroacetic Acid SCHEMBL7417558 0.84 ITGB3 (0.49) ITGB3ITGA2BF2
SCHEMBL7693853 0.84 ITGB3 (0.51) ITGB3ITGA2B
SCHEMBL7695352 0.84 ITGB3 (0.49) ITGB3ITGA2BF2
Trifluoroacetic Acid SCHEMBL7422529 0.84 ITGB3 (0.51) ITGB3ITGA2B
SCHEMBL7421961 0.83 ITGB3 (0.53) ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US claimed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP claimed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO claimed