SCHEMBL7414099

SCHEMBL7414099

Cc1c(C)c(C)c(S(=O)(=O)N[C@@H](Cc2ccc(OCCCONC(=N)N)cc2)C(=O)O)c(C)c1C

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 15/20 0.53
ITGA2B P08514 14/20 0.53
PPARG P37231 1/20 0.43
ITGAV P06756 2/20 0.42
CHRM2 P08172 1/20 0.42
SLC6A4 P31645 1/20 0.42
MMP2 P08253 1/20 0.42
MMP9 P14780 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
KCNA5 P22460 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL7417558 0.95 ITGB3 (0.49) ITGB3ITGA2BPPARGITGAVCHRM2
SCHEMBL7418575 0.89 ITGB3 (0.55) ITGB3ITGA2BITGAV
SCHEMBL7412563 0.88 AVPR1B (0.51) ITGB3ITGA2B
SCHEMBL7412450 0.88 ITGB3 (0.69) ITGB3ITGA2BPPARGITGAVCHRM2
SCHEMBL7411712 0.87 TDP1 (0.59) ITGB3ITGA2BMMP2MMP9TDP1
SCHEMBL7423110 0.87 ITGB3 (0.48) ITGB3ITGA2BPPARGITGAVMMP2
SCHEMBL7418686 0.86 ITGB1 (0.51) ITGB3ITGA2BPPARGITGAV
SCHEMBL7416684 0.86 ITGB3 (0.52) ITGB3ITGA2BITGAV
SCHEMBL7463784 0.86 ITGB3 (0.48) ITGB3ITGA2BITGAV
SCHEMBL7420817 0.86 ITGB3 (0.56) ITGB3ITGA2BITGAVCHRM2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US claimed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP claimed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO claimed