SCHEMBL7412592

SCHEMBL7412592

COc1cccc(C(CN)C(C)C)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.56
AOC3 Q16853 3/20 0.53
L3MBTL1 Q9Y468 1/20 0.49
CASR P41180 3/20 0.48
ALDH1A1 P00352 1/20 0.44
CYP3A4 P08684 1/20 0.44
CHEK1 O14757 1/20 0.42
ROCK2 O75116 1/20 0.42
RPS6KA5 O75582 1/20 0.42
MAP4K4 O95819 1/20 0.42
CHEK2 O96017 1/20 0.42
PRKCG P05129 1/20 0.42
CDK1 P06493 1/20 0.42
PRKACA P17612 1/20 0.42
RPS6KB1 P23443 1/20 0.42
CDK2 P24941 1/20 0.42
MAPK1 P28482 1/20 0.42
AKT1 P31749 1/20 0.42
AKT2 P31751 1/20 0.42
GSK3A P49840 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18320847 0.84 AOC3 (0.50) TAAR1AOC3L3MBTL1CASR
SCHEMBL18403140 0.84 AOC3 (0.50) TAAR1AOC3L3MBTL1CASR
SCHEMBL27536288 0.83 AOC3 (0.49) TAAR1AOC3L3MBTL1CASRMAPK1
SCHEMBL413321 0.82 TAAR1 (0.53) TAAR1AOC3L3MBTL1CASRALDH1A1
SCHEMBL410128 0.82 TAAR1 (0.53) TAAR1AOC3L3MBTL1CASRALDH1A1
SCHEMBL2176341 0.82 AOC3 (0.47) TAAR1AOC3L3MBTL1CASRALDH1A1
SCHEMBL16871235 0.82 AOC3 (0.47) TAAR1AOC3L3MBTL1CASRALDH1A1
SCHEMBL10245271 0.81 AOC3 (0.48) TAAR1AOC3L3MBTL1CASR
SCHEMBL9212842 0.81 AOC3 (0.51) TAAR1AOC3L3MBTL1CASRALDH1A1
SCHEMBL11081355 0.80 AOC3 (0.54) TAAR1AOC3L3MBTL1CASRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6358973-B1 FOR THERAPY OF ALLERGIC OR INFLAMMATORY DISEASE ZAMBON GROUP S.P.A. (IT) 2002-03-19 US disclosed
EP-1121353-A1 BENZAZINE DERIVATIVES AS PHOSPHODIESTERASE 4 INHIBITORS ZAMBON GROUP S.p.A. (IT) 2001-08-08 EP disclosed
WO-2000021947-A1 BENZAZINE DERIVATIVES AS PHOSPHODIESTERASE 4 INHIBITORS ZAMBON GROUP S.P.A. (IT) 2000-04-20 WO disclosed