SCHEMBL7413083

SCHEMBL7413083

Nc1ccccc1NC(=O)C1=C(O)CCc2c1nc1ccccn21

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 11/20 0.42
HDAC2 Q92769 4/20 0.42
HDAC3 O15379 3/20 0.39
MAPK1 P28482 1/20 0.39
HDAC7 Q8WUI4 2/20 0.39
HDAC9 Q9UKV0 2/20 0.39
HDAC5 Q9UQL6 2/20 0.39
HDAC4 P56524 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
NTRK1 P04629 2/20 0.39
EPHB3 P54753 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7957484 0.89 POLB (0.45) EPHB3POLB
SCHEMBL7418614 0.87 EPHB3 (0.54) MAPK1NTRK1EPHB3
SCHEMBL7959624 0.87 NPC1 (0.48) MAPK1POLB
SCHEMBL7961323 0.84 EPHB3 (0.46) NTRK1EPHB3POLB
SCHEMBL7418952 0.84 RAB9A (0.44) NTRK1
SCHEMBL7964125 0.83 NTRK1 (0.43) NTRK1EPHB3POLB
SCHEMBL7964544 0.83 KMT2A (0.42) HDAC3HDAC7HDAC9HDAC5NCOR2
SCHEMBL7420479 0.83 NTRK1 (0.43) MAPK1NTRK1EPHB3POLB
SCHEMBL7418615 0.83 KCNK3 (0.45) HDAC3HDAC7HDAC9HDAC5NCOR2
SCHEMBL7412623 0.83 IGF1R (0.45) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5639760-A USEFUL AS MUSCLE RELAXANTS, SEDATIVES, ANXIOLYTICS, ANTICONVULSANTS, AND ANTIDOTES FOR DRUG OVERDOSE MARYANOFF BRUCE E (US) 1997-06-17 US claimed
US-6218384-B1 FOR THERAPY OF ANXIETY, MUSCLE SPASMS, SLEEPLESSNESS, CONVULSIONS AND BENZODIAZEPINE OVERDOSES ORTHO-MCNEIL PHARMACEUTICAL, INC. 2001-04-17 US disclosed
US-5639760-A USEFUL AS MUSCLE RELAXANTS, SEDATIVES, ANXIOLYTICS, ANTICONVULSANTS, AND ANTIDOTES FOR DRUG OVERDOSE MARYANOFF BRUCE E (US) 1997-06-17 US disclosed
WO-1994004532-A1 3-OXO-PYRIDO(1,2-A^_)BENZIMIDAZOLE-4-CARBOXYL AND 4-OXO-AZEPINO(1,2-A^_)BENZIMIDAZOLE-5-CARBOXYL DERIVATIVES USEFUL IN TREATING CENTRAL NERVOUS SYSTEM DISORDERS MCNEILAB, INC. (US) 1994-03-03 WO disclosed