SCHEMBL7959624

SCHEMBL7959624

Cc1ccccc1NC(=O)C1=C(O)CCc2c1nc1ccccn21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
ALDH1A1 P00352 3/20 0.48
HPGD P15428 3/20 0.48
TP53 P04637 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
MAPK1 P28482 3/20 0.43
POLB P06746 2/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
GAA P10253 4/20 0.41
KDM4E B2RXH2 4/20 0.41
LMNA P02545 3/20 0.41
HTT P42858 3/20 0.41
MAPT P10636 2/20 0.41
GFER P55789 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
PKM P14618 3/20 0.40
PKLR P30613 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7418614 0.87 EPHB3 (0.54) NPC1RAB9AHPGDMAPK1
SCHEMBL7413083 0.87 HDAC1 (0.42) MAPK1POLB
SCHEMBL7957484 0.87 POLB (0.45) POLB
SCHEMBL7961323 0.84 EPHB3 (0.46) NPC1RAB9ATP53SMN1; SMN2POLB
SCHEMBL7418952 0.84 RAB9A (0.44) NPC1RAB9ASMN1; SMN2KMT2AGAA
SCHEMBL7949786 0.84 NTRK1 (0.46) NPC1RAB9AALDH1A1HPGDPOLB
SCHEMBL7420479 0.83 NTRK1 (0.43) NPC1RAB9AALDH1A1SMN1; SMN2MAPK1
SCHEMBL7964125 0.83 NTRK1 (0.43) NPC1RAB9AALDH1A1HPGDSMN1; SMN2
SCHEMBL7964322 0.82 NTRK1 (0.43) NPC1RAB9AALDH1A1HPGDMAPK1
SCHEMBL7959855 0.82 LMNA (0.44) NPC1RAB9AHPGDTP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5639760-A USEFUL AS MUSCLE RELAXANTS, SEDATIVES, ANXIOLYTICS, ANTICONVULSANTS, AND ANTIDOTES FOR DRUG OVERDOSE MARYANOFF BRUCE E (US) 1997-06-17 US claimed
US-6218384-B1 FOR THERAPY OF ANXIETY, MUSCLE SPASMS, SLEEPLESSNESS, CONVULSIONS AND BENZODIAZEPINE OVERDOSES ORTHO-MCNEIL PHARMACEUTICAL, INC. 2001-04-17 US disclosed
US-5639760-A USEFUL AS MUSCLE RELAXANTS, SEDATIVES, ANXIOLYTICS, ANTICONVULSANTS, AND ANTIDOTES FOR DRUG OVERDOSE MARYANOFF BRUCE E (US) 1997-06-17 US disclosed