SCHEMBL741362

SCHEMBL741362

CCOC(=O)C1CCC(NC(=O)c2cc3cc(F)ccc3[nH]2)(C(=O)OC(C)(C)C)C(N)C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MLLT1 Q03111 1/20 0.40
RAB9A P51151 3/20 0.40
NPC1 O15118 2/20 0.40
POLB P06746 1/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
ATM Q13315 1/20 0.39
SMYD3 Q9H7B4 1/20 0.39
PYGL P06737 4/20 0.37
GHSR Q92847 1/20 0.36
METAP2 P50579 2/20 0.36
CNR1 P21554 1/20 0.35
PYGM P11217 1/20 0.35
RXFP1 Q9HBX9 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
KCNA6 P17658 1/20 0.34
KCNA3 P22001 1/20 0.34
KCNA4 P22459 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL739706 0.91 KMT2A (0.50) RAB9AMEN1KMT2AATMSMYD3
SCHEMBL741538 0.80 SMYD3 (0.46) SMYD3PYGL
SCHEMBL743763 0.80 SMYD3 (0.46) SMYD3PYGL
SCHEMBL740808 0.78 F10 (0.44) SMYD3PYGL
SCHEMBL739377 0.78 F10 (0.44) SMYD3PYGL
SCHEMBL765158 0.76 MLLT1 (0.47) MLLT1RAB9ANPC1POLBMEN1
SCHEMBL740438 0.76 SMYD3 (0.45) SMYD3PYGL
SCHEMBL741757 0.75 SMYD3 (0.46) SMYD3PYGL
SCHEMBL741108 0.75 SMYD3 (0.44) SMYD3PYGL
SCHEMBL11888215 0.72 MLLT1 (0.67) MLLT1RAB9ANPC1POLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2431370-A1 Monoacylated 1,2-diaminocycloalkanes DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2012-03-21 EP disclosed
US-7935824-B2 Ethylenediamine derivatives DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2011-05-03 US disclosed