SCHEMBL740808

SCHEMBL740808

CN(C)C(=O)C1CCC(NC(=O)c2cc3cc(Cl)ccc3[nH]2)(C(=O)OC(C)(C)C)C(N)C1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
F10 P00742 6/20 0.44
SMYD3 Q9H7B4 1/20 0.44
PYGL P06737 10/20 0.43
F2 P00734 1/20 0.42
PLAT P00750 1/20 0.42
CYP51A1 Q16850 1/20 0.42
IDO1 P14902 1/20 0.42
HRH4 Q9H3N8 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741538 0.92 SMYD3 (0.46) SMYD3PYGLCYP51A1IDO1HRH4
SCHEMBL743763 0.92 SMYD3 (0.46) F10SMYD3PYGLCYP51A1IDO1
SCHEMBL739377 0.89 F10 (0.44) F10SMYD3PYGLCYP51A1IDO1
SCHEMBL739706 0.88 KMT2A (0.50) SMYD3PYGLCYP51A1IDO1
SCHEMBL741757 0.87 SMYD3 (0.46) SMYD3PYGLCYP51A1IDO1
SCHEMBL740438 0.86 SMYD3 (0.45) SMYD3PYGLCYP51A1IDO1HRH4
SCHEMBL741108 0.85 SMYD3 (0.44) SMYD3PYGLCYP51A1IDO1HRH4
SCHEMBL743062 0.84 F10 (0.32) F10
SCHEMBL743324 0.81 F10 (0.46) F10
SCHEMBL741362 0.78 MLLT1 (0.40) SMYD3PYGL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2431370-A1 Monoacylated 1,2-diaminocycloalkanes DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2012-03-21 EP disclosed
US-7935824-B2 Ethylenediamine derivatives DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2011-05-03 US disclosed