SCHEMBL743763

SCHEMBL743763

CC(C)(C)OC(=O)C1(NC(=O)c2cc3cc(Cl)ccc3[nH]2)CCC(C(=O)O)CC1N

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.46
CYP51A1 Q16850 1/20 0.43
IDO1 P14902 6/20 0.43
PYGL P06737 9/20 0.42
F10 P00742 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741538 0.93 SMYD3 (0.46) SMYD3CYP51A1IDO1PYGL
SCHEMBL740808 0.92 F10 (0.44) SMYD3CYP51A1IDO1PYGLF10
SCHEMBL739377 0.91 F10 (0.44) SMYD3CYP51A1IDO1PYGLF10
SCHEMBL739706 0.90 KMT2A (0.50) SMYD3CYP51A1IDO1PYGL
SCHEMBL741757 0.88 SMYD3 (0.46) SMYD3CYP51A1IDO1PYGL
SCHEMBL740438 0.87 SMYD3 (0.45) SMYD3CYP51A1IDO1PYGL
SCHEMBL741108 0.86 SMYD3 (0.44) SMYD3CYP51A1IDO1PYGL
SCHEMBL741362 0.80 MLLT1 (0.40) SMYD3PYGL
SCHEMBL743062 0.76 F10 (0.32) F10
SCHEMBL742116 0.74 SMYD3 (0.47) SMYD3PYGLF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2431370-A1 Monoacylated 1,2-diaminocycloalkanes DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2012-03-21 EP disclosed
US-7935824-B2 Ethylenediamine derivatives DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2011-05-03 US disclosed