SCHEMBL7414541

SCHEMBL7414541

Cc1ccccc1S(=O)(=O)OCC1CCN1C(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 4/20 0.41
NR1H3 Q13133 3/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
STS P08842 1/20 0.40
TGFBR1 P36897 1/20 0.40
HCRTR2 O43614 1/20 0.40
LMNA P02545 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
GPR119 Q8TDV5 1/20 0.39
KDM4E B2RXH2 1/20 0.38
PKM P14618 1/20 0.38
KDM1A O60341 1/20 0.38
CCR5 P51681 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7667825 1.00 NR1H2 (0.41) NR1H2NR1H3MEN1KMT2ASTS
SCHEMBL7407543 1.00 NR1H2 (0.41) NR1H2NR1H3MEN1KMT2ASTS
SCHEMBL7734440 0.93 MEN1 (0.46) NR1H2NR1H3MEN1KMT2ASTS
SCHEMBL28433249 0.93 MEN1 (0.46) NR1H2NR1H3MEN1KMT2ASTS
SCHEMBL345694 0.83 GPR119 (0.44) NR1H2NR1H3MEN1KMT2ASTS
SCHEMBL2186144 0.83 GPR119 (0.44) NR1H2NR1H3MEN1KMT2ASTS
SCHEMBL345693 0.83 GPR119 (0.44) NR1H2NR1H3MEN1KMT2ASTS
SCHEMBL1879006 0.83 TGFBR1 (0.52) STSTGFBR1GPR119KDM4EPKM
SCHEMBL7414415 0.83 NR1H2 (0.39) NR1H2NR1H3MEN1KMT2ASTS
SCHEMBL7414543 0.81 STS (0.53) NR1H2NR1H3KMT2ASTSHCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0950057-B1 3-PYRIDYL ENANTIOMERS AND THEIR USE AS ANALGESICS ABBOTT LAB (US) 2002-11-13 EP disclosed
US-6403575-B1 ANTI-INFLAMMATORIES ABBOTT LABORATORIES 2002-06-11 US disclosed
EP-1047690-A1 HETEROCYCLIC ETHER AND THIOETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 2000-11-02 EP disclosed
US-6133253-A NEURONAL CELL DEATH PREVENTORS AND ANTI-INFLAMMATORIES ABBOTT LABORATORIES (US) 2000-10-17 US disclosed
WO-1999032480-A1 HETEROCYCLIC ETHER AND THIOETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1999-07-01 WO disclosed