SCHEMBL7414714

SCHEMBL7414714

Cc1ccc2[nH]c(N3CCCN(C)CC3)nc2c1OC(N)=O

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
HRH4 Q9H3N8 3/20 0.39
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
GFER P55789 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7411450 0.87 PARP1 (0.39) PARP1HRH4
SCHEMBL6873048 0.82 PARP1 (0.47) PARP1HRH4
SCHEMBL6874969 0.77 PARP1 (0.51) PARP1HRH4
SCHEMBL5621000 0.76 PARP1 (0.68) PARP1
SCHEMBL7411210 0.75 PARP1 (0.37) PARP1
SCHEMBL7410126 0.74 NPY5R (0.44) PARP1NPC1RAB9AHRH4
SCHEMBL7415578 0.74 PIM1 (0.40) PARP1HRH4
SCHEMBL7408313 0.74 NPC1 (0.52) PARP1NPC1RAB9AHRH4
SCHEMBL7417446 0.73 HTR3A (0.40) PARP1
SCHEMBL6314907 0.72 PARP1 (0.36) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed