SCHEMBL7417446

SCHEMBL7417446

CCc1ccc2[nH]c(N3CCNCC3)nc2c1OC(N)=O

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.40
PARP1 P09874 14/20 0.40
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
NAMPT P43490 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7415578 0.96 PIM1 (0.40) HTR3APARP1ITGB3ITGA2B
SCHEMBL7038510 0.78 KCNH2 (0.37) HTR3APARP1ITGB3ITGA2BNAMPT
SCHEMBL6869623 0.78 PARP1 (0.49) HTR3APARP1NAMPT
SCHEMBL7045004 0.75 PIM1 (0.38) HTR3APARP1ITGB3ITGA2B
SCHEMBL6864445 0.74 PARP1 (0.46) HTR3APARP1
SCHEMBL7414570 0.74 HTR3A (0.40) HTR3APARP1ITGB3ITGA2BNAMPT
SCHEMBL7410717 0.74 PARP1 (0.39) PARP1
SCHEMBL7411360 0.73 PARP1 (0.56) PARP1
SCHEMBL7411450 0.73 PARP1 (0.39) PARP1
SCHEMBL7414714 0.73 PARP1 (0.40) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed