SCHEMBL7414927

SCHEMBL7414927

O=C(c1ccc(F)cc1Br)N1C=C2CC=CN2Cc2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 9/20 0.41
AVPR1A P37288 6/20 0.41
OXTR P30559 2/20 0.41
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
P2RX7 Q99572 3/20 0.33
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32
TAS1R2 Q8TE23 1/20 0.32
HSP90B1 P14625 2/20 0.32
TRAP1 Q12931 2/20 0.32
GAA P10253 1/20 0.32
HTT P42858 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7422025 0.90 AVPR2 (0.42) AVPR2AVPR1AOXTRP2RX7TAS1R3
SCHEMBL7421754 0.88 AVPR2 (0.50) AVPR2AVPR1AOXTRNPC1P2RX7
SCHEMBL7417501 0.86 AVPR2 (0.40) AVPR2AVPR1AOXTRMAPTP2RX7
SCHEMBL7420622 0.81 AVPR2 (0.43) AVPR2AVPR1AOXTR
SCHEMBL7421267 0.76 AVPR2 (0.38) AVPR2AVPR1AOXTR
SCHEMBL2313462 0.76 HSD17B3 (0.32) MAPTALDH1A1
SCHEMBL7549935 0.75 BCAT2 (0.34) AVPR2AVPR1AOXTRNPC1MAPT
SCHEMBL7638228 0.75 AVPR2 (0.57) AVPR2AVPR1AOXTR
SCHEMBL4394751 0.72 AVPR2 (0.48) AVPR2AVPR1AOXTR
SCHEMBL7422271 0.71 AVPR2 (0.52) AVPR2AVPR1AOXTRP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000062-A1 TRICYCLIC VASOPRESSIN AGONISTS AMERICAN HOME PRODUCTS CORPORATION (US) 2000-05-17 EP disclosed
WO-1999006409-A1 TRICYCLIC VASOPRESSIN AGONISTS AMERICAN HOME PRODUCTS CORPORATION (US) 1999-02-11 WO disclosed