SCHEMBL7415633

SCHEMBL7415633

ClCc1ccc(Cl)c(Cl)c1.c1ccc(P(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.46
TDP1 Q9NUW8 2/20 0.44
CYP3A4 P08684 1/20 0.44
IDO1 P14902 3/20 0.44
PNMT P11086 2/20 0.41
TAAR1 Q96RJ0 1/20 0.41
SLC6A2 P23975 2/20 0.41
SLC6A4 P31645 2/20 0.41
SLC6A3 Q01959 2/20 0.41
CCR2 P41597 3/20 0.39
PLAAT3 P53816 1/20 0.39
PLAAT5 Q96KN8 1/20 0.39
PLAAT2 Q9NWW9 1/20 0.39
PLAAT4 Q9UL19 1/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
PTPRG P23470 1/20 0.39
PLA2G1B P04054 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4962307 0.84 SIGMAR1 (0.45) SIGMAR1TDP1CYP3A4IDO1PNMT
SCHEMBL11411021 0.83 PNMT (0.41) SIGMAR1CYP3A4IDO1PNMTTAAR1
SCHEMBL29494831 0.82 IDO1 (0.61) SIGMAR1IDO1PNMTTAAR1SLC6A2
SCHEMBL407334 0.82 IDO1 (0.61) SIGMAR1IDO1PNMTTAAR1SLC6A2
SCHEMBL22871613 0.80 CYP3A4 (0.57) TDP1CYP3A4KMT2ATSHR
Ammonia Solution, Strong SCHEMBL14485188 0.80 IDO1 (0.58) SIGMAR1IDO1PNMTTAAR1SLC6A2
SCHEMBL16618385 0.80 IDO1 (0.58) SIGMAR1IDO1PNMTTAAR1SLC6A2
SCHEMBL6201046 0.79 TDP1 (0.50) SIGMAR1TDP1CYP3A4IDO1PLAAT3
Hydrochloric Acid SCHEMBL5143704 0.78 CYP3A4 (0.55) TDP1CYP3A4KMT2ATSHR
(Chloromethyl)Benzene SCHEMBL304085 0.78 CYP3A4 (0.60) SIGMAR1TDP1CYP3A4IDO1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6013656-A PSYCHOLOGICAL DISORDERS; GASTROINTESTINAL DISORDERS; NERVOUSSYSTEM DISORDERS WARNER-LAMBERT COMPANY (US) 2000-01-11 US disclosed
US-5849760-A 2-(arylalkenyl)azacycloalkane derivatives as ligands for sigma receptors INSTITUT DE RECHERCHE JOUVEINAL (FR) 1998-12-15 US disclosed
US-4187300-A Use of phosphonium salts in treatment of African trypanosomiasis THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE ARMY (US) 1980-02-05 US disclosed