Acetic Acid

Acetic Acid

SCHEMBL7415684

CC(=O)O.CCOC(=O)C[C@H](NC(=O)N[C@H]1CCN(c2ccc(C(=N)N)cc2)C1=O)c1ccccc1

nearest known ligand 0.64

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Known targets — ChEMBL curated mechanism

ADRA2AADRA2BADRA2CADRB2AGTR1AVPR1AAVPR1BAVPR2BDKRB2CALCRCHRNA3CHRNB4ESR1ESR2GHSRGNRHRGSC1HSPA8MALT1MC1RMC4RNOS1NOS2NOS3OPRK1OXTRRAMP1RAMP2RAMP3SCN5ASSTR1SSTR2SSTR3SSTR4SSTR5dacAdacBdacCfolPftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Acetic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 13/20 0.64
ITGA2B P08514 13/20 0.64
F10 P00742 6/20 0.47
F2 P00734 5/20 0.47
LMNA P02545 1/20 0.42
PRSS1 P07477 6/20 0.41
PRSS2 P07478 5/20 0.41
PRSS3 P35030 5/20 0.41
FPR1 P21462 1/20 0.39
FPR2 P25090 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7419223 0.89 ITGB3 (0.53) ITGB3ITGA2BF10F2LMNA
Acetic Acid SCHEMBL7414160 0.88 ITGB3 (0.68) ITGB3ITGA2BF10F2PRSS1
SCHEMBL8115160 0.86 ITGB3 (0.71) ITGB3ITGA2BF10F2PRSS1
SCHEMBL8108543 0.86 ITGB3 (0.71) ITGB3ITGA2BF10F2PRSS1
SCHEMBL7424541 0.85 ITGB3 (0.51) ITGB3ITGA2BF10F2FPR1
SCHEMBL7411896 0.84 ITGB3 (0.47) ITGB3ITGA2BLMNAFPR1FPR2
SCHEMBL7417192 0.84 ITGB3 (0.67) ITGB3ITGA2BF10F2PRSS1
SCHEMBL7421976 0.84 ITGB3 (0.51) ITGB3ITGA2BF10F2LMNA
SCHEMBL7417201 0.84 ITGB3 (0.67) ITGB3ITGA2BF10F2PRSS1
SCHEMBL7417196 0.84 ITGB3 (0.67) ITGB3ITGA2BF10F2PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0796245-B1 PROCESS FOR THE PREPARATION OF AMIDINO PHENYL PYRROLIDINE BETA-ALANINE UREA ANALOGS SEARLE & CO (US) 2000-07-26 EP disclosed
US-5659063-A AMINE-BLOCKED METHIONINE ANALOG CYCLIZABLE TO A LACTAM IN NONVOLATILE OR NONTOXIC REAGENTS; ANTITHROMBOTIC AGENTS G. D. SEARLE & CO. (US) 1997-08-19 US disclosed
US-5610296-A CHEMICAL INTERMEDIATES OF ANTITHROMBOTICS G. D. SEARLE & CO. (US) 1997-03-11 US disclosed
WO-1996017827-A1 PROCESS FOR THE PREPARATION OF AMIDINO PHENYL PYRROLIDINE β-ALANINE UREA ANALOGS G.D. SEARLE & CO. (US) 1996-06-13 WO disclosed
US-5484946-A CYCLIZATION AND DEHYDRATION A METHIONINE DERIVATIVE G. D. SEARLE & CO. (US) 1996-01-16 US disclosed