SCHEMBL7415931

SCHEMBL7415931

CC(=O)Nc1ccc(C(=O)O)c2c1C=CCO2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.42
HSD17B10 Q99714 4/20 0.42
CASP1 P29466 1/20 0.36
ALDH1A1 P00352 4/20 0.35
ALOX15 P16050 1/20 0.35
POLB P06746 3/20 0.35
CYP2C19 P33261 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MTNR1A P48039 2/20 0.33
KMT2A Q03164 2/20 0.33
MAPT P10636 1/20 0.33
MTNR1B P49286 1/20 0.33
NEU3 Q9UQ49 1/20 0.33
MEN1 O00255 1/20 0.33
HPGD P15428 2/20 0.32
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
MAOA P21397 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7333342 0.86 SMN1; SMN2 (0.40) KDM4EHSD17B10CASP1ALDH1A1ALOX15
SCHEMBL7333144 0.75 KDM4E (0.37) KDM4EHSD17B10ALDH1A1ALOX15POLB
SCHEMBL5760894 0.75 ALB (0.33) CASP1NPC1SMN1; SMN2CYP1A2
SCHEMBL7396214 0.75 KDM4E (0.47) KDM4EHSD17B10CASP1ALDH1A1ALOX15
SCHEMBL1435852 0.71 HSD17B10 (0.48) KDM4EHSD17B10CASP1ALDH1A1ALOX15
SCHEMBL2965600 0.69 HSD17B10 (0.46) KDM4EHSD17B10CASP1ALDH1A1ALOX15
SCHEMBL5759463 0.69 TSHR (0.37) KDM4EHSD17B10CASP1ALDH1A1POLB
SCHEMBL5763798 0.69 GYS1 (0.35) CASP1NPC1SMN1; SMN2CYP1A2
SCHEMBL27974832 0.67 PARP1 (0.48) KDM4EHSD17B10ALDH1A1POLBCYP2C19
SCHEMBL7333041 0.66 KDM4E (0.51) KDM4EHSD17B10ALDH1A1POLBCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127379-A TREATING IRRITABLE BOWEL SYNDROME, URINARY INCONTINENCE, ATRIAL ARRHYTHMIA OR STROKE SMITHKLINE BEECHAM P.L.C. (GB) 2000-10-03 US disclosed
EP-0625149-A1 BENZOPYRAN, BENZOTHIOPYRAN AND BENZOFURAN DERIVATIVES AS 5-HT4 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-11-23 EP disclosed
WO-1993016072-A1 BENZOPYRAN, BENZOTHIOPYRAN AND BENZOFURAN DERIVATIVES AS 5-HT4 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1993-08-19 WO disclosed