SCHEMBL7416213

SCHEMBL7416213

CC(C)CC(NC(=O)C(C)Oc1cccc2ccccc12)C(=O)[C@H](C=O)C(N)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 6/20 0.52
CASP1 P29466 5/20 0.52
CASP7 P55210 5/20 0.52
CASP6 P55212 5/20 0.52
CASP8 Q14790 5/20 0.52
PSMB5 P28074 1/20 0.45
PTGS2 P35354 1/20 0.43
BCL2L1 Q07817 1/20 0.43
NTSR1 P30989 1/20 0.42
ANPEP P15144 2/20 0.41
MME P08473 1/20 0.38
ACE P12821 1/20 0.38
CPA1 P15085 1/20 0.38
ACE2 Q9BYF1 1/20 0.38
CARM1 Q86X55 1/20 0.38
PRMT6 Q96LA8 1/20 0.38
SLC1A3 P43003 1/20 0.38
SLC1A2 P43004 1/20 0.38
SLC1A1 P43005 1/20 0.38
FNTA P49354 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7622869 1.00 CASP3 (0.52) CASP3CASP1CASP7CASP6CASP8
SCHEMBL7627735 0.88 CASP3 (0.57) CASP3CASP1CASP7CASP6CASP8
SCHEMBL7619325 0.88 CASP3 (0.57) CASP3CASP1CASP7CASP6CASP8
SCHEMBL7420035 0.88 CASP3 (0.57) CASP3CASP1CASP7CASP6CASP8
SCHEMBL7413527 0.88 CASP3 (0.57) CASP3CASP1CASP7CASP6CASP8
SCHEMBL7467278 0.86 CASP3 (0.53) CASP3CASP1CASP7CASP6CASP8
SCHEMBL7672483 0.82 ANPEP (0.48) PSMB5NTSR1ANPEPMMEACE
SCHEMBL7625305 0.82 ANPEP (0.48) PSMB5NTSR1ANPEPMMEACE
SCHEMBL5488516 0.80 CASP3 (0.55) CASP3CASP1CASP7CASP6CASP8
SCHEMBL5971546 0.73 CAPN1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1123272-A1 (SUBSTITUTED)ACYL DIPEPTIDYL INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE PROTEASES Idun Pharmaceuticals, Inc. (US) 2001-08-16 EP disclosed
WO-2000023421-A1 (SUBSTITUTED)ACYL DIPEPTIDYL INHIBITORS OF THE ICE/ced-3 FAMILY OF CYSTEINE PROTEASES IDUN PHARMACEUTICALS, INC. (US) 2000-04-27 WO disclosed