SCHEMBL7420035

SCHEMBL7420035

CC(C)C[C@H](NC(=O)C(CCC(=O)O)Oc1cccc2ccccc12)C(=O)[C@H](C=O)C(N)C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 5/20 0.57
CASP1 P29466 4/20 0.57
CASP7 P55210 4/20 0.57
CASP6 P55212 4/20 0.57
CASP8 Q14790 4/20 0.57
PSMB5 P28074 1/20 0.48
ERAP2 Q6P179 5/20 0.43
IL1RN P18510 4/20 0.40
ERAP1 Q9NZ08 3/20 0.40
BCL2L1 Q07817 1/20 0.38
NTSR1 P30989 1/20 0.38
ANPEP P15144 1/20 0.38
MMP3 P08254 1/20 0.36
FOLH1 Q04609 4/20 0.36
BACE1 P56817 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7627735 1.00 CASP3 (0.57) CASP3CASP1CASP7CASP6CASP8
SCHEMBL7413527 1.00 CASP3 (0.57) CASP3CASP1CASP7CASP6CASP8
SCHEMBL7619325 1.00 CASP3 (0.57) CASP3CASP1CASP7CASP6CASP8
SCHEMBL7416213 0.88 CASP3 (0.52) CASP3CASP1CASP7CASP6CASP8
SCHEMBL7622869 0.88 CASP3 (0.52) CASP3CASP1CASP7CASP6CASP8
SCHEMBL5494420 0.82 CASP1 (0.60) CASP3CASP1CASP7CASP6CASP8
SCHEMBL5496384 0.82 CASP1 (0.60) CASP3CASP1CASP7CASP6CASP8
SCHEMBL14598380 0.82 CASP1 (0.60) CASP3CASP1CASP7CASP6CASP8
SCHEMBL14598379 0.82 CASP1 (0.60) CASP3CASP1CASP7CASP6CASP8
SCHEMBL7467278 0.82 CASP3 (0.53) CASP3CASP1CASP7CASP6CASP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1123272-A1 (SUBSTITUTED)ACYL DIPEPTIDYL INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE PROTEASES Idun Pharmaceuticals, Inc. (US) 2001-08-16 EP disclosed
WO-2000023421-A1 (SUBSTITUTED)ACYL DIPEPTIDYL INHIBITORS OF THE ICE/ced-3 FAMILY OF CYSTEINE PROTEASES IDUN PHARMACEUTICALS, INC. (US) 2000-04-27 WO disclosed