SCHEMBL7416243

SCHEMBL7416243

N#Cc1cc(CN2CC[C@H](N)C2=O)cs1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.36
F2 P00734 2/20 0.33
F10 P00742 2/20 0.33
PLG P00747 1/20 0.33
PLAT P00750 1/20 0.33
PROC P04070 1/20 0.33
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
MAPT P10636 1/20 0.32
APEX1 P27695 1/20 0.32
S100A9 P06702 1/20 0.32
TNKS O95271 1/20 0.30
TNKS2 Q9H2K2 1/20 0.30
FNTA P49354 3/20 0.30
FNTB P49356 3/20 0.30
PGGT1B P53609 3/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7422788 1.00 TRPA1 (0.36) TRPA1F2F10PLGPLAT
Hydrochloric Acid SCHEMBL2326785 0.99 TRPA1 (0.35) TRPA1F2F10PLGPLAT
Hydrochloric Acid SCHEMBL2326780 0.99 TRPA1 (0.35) TRPA1F2F10PLGPLAT
SCHEMBL7421074 0.85 TRPA1 (0.37) TRPA1F2F10PLGPLAT
SCHEMBL27493529 0.84 TRPA1 (0.36) TRPA1F2F10PLGPLAT
SCHEMBL7416241 0.83 TRPA1 (0.35) TRPA1F2F10PLGPLAT
SCHEMBL7423307 0.81 F10 (0.39) TRPA1F2F10CYP3A4S100A9
SCHEMBL27494330 0.79 TRPA1 (0.35) TRPA1F2F10PLGPLAT
SCHEMBL2325183 0.77 F10 (0.44) F2F10PLGPROC
SCHEMBL7424915 0.76 DPP4 (0.33) F2F10CYP3A4TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853618-A4 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHONE POULENC RORER PHARMA (US) 2000-03-15 EP disclosed
US-6034093-A Substituted sulfonic acid N-[(aminoiminomethyl)phenylalkyl]-azaheterocyclylamide compounds RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 2000-03-07 US disclosed
EP-0853618-A1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1998-07-22 EP disclosed
WO-1996040679-A1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N-[(AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHÔNE-POULENC RORER PHARMACEUTICALS INC. (US) 1996-12-19 WO disclosed