SCHEMBL7416503

SCHEMBL7416503

NC(=O)C1C=C(Cl)N(CCc2ccccc2)c2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.47
KDM4E B2RXH2 1/20 0.47
PARK7 Q99497 5/20 0.43
ADRA1D P25100 1/20 0.40
ALDH2 P05091 2/20 0.40
ALDH3A1 P30838 2/20 0.40
PKM P14618 1/20 0.39
GSK3A P49840 1/20 0.38
GSK3B P49841 1/20 0.38
MGLL Q99685 1/20 0.38
SIRT1 Q96EB6 1/20 0.37
PARP1 P09874 1/20 0.37
PARP2 Q9UGN5 1/20 0.37
CACNA1G O43497 1/20 0.37
CACNA1H O95180 1/20 0.37
CACNA1I Q9P0X4 1/20 0.37
ALOX12 P18054 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29385380 0.69 ALDH1A1 (0.63) ALDH1A1KDM4EPARK7ALDH2ALDH3A1
SCHEMBL2823271 0.67 ALDH1A1 (0.59) ALDH1A1KDM4EPARK7ALDH2ALDH3A1
SCHEMBL3859755 0.62 RXFP1 (0.49) ALDH1A1KDM4EALDH2ALDH3A1GSK3A
SCHEMBL11146494 0.61 GRM2 (0.52) ALDH1A1PKM
SCHEMBL22235758 0.61 ALDH1A1 (0.60) ALDH1A1KDM4EPARK7ALDH2ALDH3A1
SCHEMBL23633187 0.61 FFAR1 (0.58) ALDH1A1
SCHEMBL8066978 0.61 KDM4E (0.69) ALDH1A1KDM4EPARK7ALDH2ALDH3A1
Hydrochloric Acid SCHEMBL28290331 0.60 OPRM1 (0.51)
Urea SCHEMBL2006220 0.60 FFAR1 (0.62) ALDH1A1
Carbamic Acid SCHEMBL2222080 0.60 FFAR1 (0.62) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0983243-A1 NOVEL QUINOLINE- AND NAPHTHALENECARBOXAMIDES, PHARMACEUTICAL COMPOSITIONS AND METHODS OF INHIBITING CALPAIN SMITHKLINE BEECHAM CORPORATION (US) 2000-03-08 EP disclosed
WO-1998041506-A1 NOVEL QUINOLINE- AND NAPHTHALENECARBOXAMIDES, PHARMACEUTICAL COMPOSITIONS AND METHODS OF INHIBITING CALPAIN SMITHKLINE BEECHAM CORPORATION (US) 1998-09-24 WO disclosed