SCHEMBL7416770

SCHEMBL7416770

CC(=O)NC(C(=O)Nc1nc(Cl)ccc1OC[C@H]1CCCN1C)c1nc(Cl)ccc1OC(C)[C@@H]1CCCN1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 4/20 0.38
CHRNA4 P43681 4/20 0.38
CHRNA7 P36544 2/20 0.38
IRAK4 Q9NWZ3 1/20 0.36
CHRNB4 P30926 4/20 0.35
CHRNA3 P32297 4/20 0.35
CHRNB1 P11230 2/20 0.35
CHRNB3 Q05901 2/20 0.35
ATR Q13535 2/20 0.33
CHRNA5 P30532 1/20 0.33
MCHR1 Q99705 2/20 0.33
CHRM3 P20309 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7407029 0.93 CHRNA3 (0.35) CHRNB2CHRNA4CHRNA7IRAK4CHRNB4
SCHEMBL7414940 0.83 IRAK4 (0.32) IRAK4
SCHEMBL7409555 0.79 CHRNA3 (0.41) CHRNB2CHRNA4IRAK4CHRNB4CHRNA3
SCHEMBL7413430 0.77 CHRNB2 (0.38) CHRNB2CHRNA4CHRNA7IRAK4CHRNB4
SCHEMBL7411849 0.76 MAPK1 (0.32)
SCHEMBL7414715 0.74 IRAK4 (0.41) CHRNB2CHRNA4CHRNA7IRAK4CHRNB4
SCHEMBL7417404 0.68 IRAK4 (0.42) CHRNB2CHRNA4IRAK4CHRNB4CHRNA3
SCHEMBL7408472 0.68 CHRNB4 (0.42) CHRNB2CHRNA4CHRNA7IRAK4CHRNB4
SCHEMBL7404130 0.67 IRAK4 (0.41) CHRNB2CHRNA4IRAK4CHRNB4CHRNA3
SCHEMBL7417095 0.65 IRAK4 (0.37) CHRNB2CHRNA4IRAK4CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047690-A1 HETEROCYCLIC ETHER AND THIOETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 2000-11-02 EP disclosed
WO-1999032480-A1 HETEROCYCLIC ETHER AND THIOETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1999-07-01 WO disclosed