SCHEMBL7416778

SCHEMBL7416778

O[CH]c1cc2ccccc2s1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.64
MGLL Q99685 1/20 0.48
BCL2L1 Q07817 1/20 0.47
GSK3B P49841 1/20 0.46
TUBB4A P04350 2/20 0.45
TUBB P07437 2/20 0.45
TUBA3C P0DPH7 2/20 0.45
TUBA1B P68363 2/20 0.45
TUBA4A P68366 2/20 0.45
TUBB4B P68371 2/20 0.45
TUBB3 Q13509 2/20 0.45
TUBB2A Q13885 2/20 0.45
TUBB8 Q3ZCM7 2/20 0.45
TUBA3E Q6PEY2 2/20 0.45
TUBA1A Q71U36 2/20 0.45
TUBA1C Q9BQE3 2/20 0.45
TUBB6 Q9BUF5 2/20 0.45
TUBB2B Q9BVA1 2/20 0.45
TUBB1 Q9H4B7 2/20 0.45
APP P05067 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2902480 0.80 CYP2A6 (0.67) CYP2A6MGLLBCL2L1GSK3BTUBB4A
SCHEMBL27556684 0.78 CYP2A6 (0.64) CYP2A6MGLLBCL2L1GSK3BTUBB4A
SCHEMBL1567141 0.78 CYP2A6 (0.64) CYP2A6MGLLBCL2L1GSK3BTUBB4A
SCHEMBL27644653 0.78 CYP2A6 (0.64) CYP2A6MGLLBCL2L1GSK3BTUBB4A
SCHEMBL56884 0.78 CYP2A6 (1.00) CYP2A6MGLLBCL2L1GSK3BTUBB4A
SCHEMBL12884253 0.78 CYP2A6 (0.64) CYP2A6MGLLBCL2L1GSK3BTUBB4A
SCHEMBL29629031 0.78 CYP2A6 (1.00) CYP2A6MGLLBCL2L1GSK3BTUBB4A
SCHEMBL1567214 0.78 CYP2A6 (0.64) CYP2A6MGLLBCL2L1GSK3BTUBB4A
SCHEMBL8996544 0.78 CYP2A6 (0.64) CYP2A6MGLLBCL2L1GSK3BTUBB4A
SCHEMBL7079637 0.78 CYP2A6 (0.64) CYP2A6MGLLBCL2L1GSK3BTUBB4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 78 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4839352-A ANTIBIOTICS MERCK & CO., INC. (US) 1989-06-13 US claimed
US-4342869-A Cephalosporin antibiotics MERCK & CO., INC. (US) 1982-08-03 US claimed
US-4338437-A Cephalosporin antibiotics MERCK & CO., INC. (US) 1982-07-06 US claimed
US-4338438-A Cephalosporin antibiotics MERCK & CO., INC. (US) 1982-07-06 US claimed
US-4310459-A Process for producing carbamoyl substituted penams and carbamoyl substituted cephams from penicillin sulfoxide esters BRISTOL-MYERS COMPANY (US) 1982-01-12 US claimed
US-4297488-A 7-α-Methoxy cephalosporins MERCK & CO., INC. (US) 1981-10-27 US claimed
US-4957912-A ANTIBIOTICS MERCK & CO., INC. (US) 1990-09-18 US disclosed
US-4891370-A ELASTASE INHIBITORS MERCK & CO., INC. (US) 1990-01-02 US disclosed
US-4847247-A ELASTASE INHIBITORS MERCK & CO., INC. (US) 1989-07-11 US disclosed
US-4845088-A ANTIINFLAMMATORY, ANTIDEGENERATIVE AGENTS MERCK & CO., INC. (US) 1989-07-04 US disclosed
US-4839352-A ANTIBIOTICS MERCK & CO., INC. (US) 1989-06-13 US disclosed
US-4797396-A INHIBITION OF ELASTASE, ANTIBIOTICS MERCK & CO., INC. (US) 1989-01-10 US disclosed
US-4717722-A ELASTASE INHIBITORS MERCK & CO., INC. (US) 1988-01-05 US disclosed
US-4071529-A Derivatives of 6-aminopenicillanic acid MERCK & CO., INC. (US) 1978-01-31 US disclosed
US-4064344-A ANTIBIOTIC MERCK & CO., INC. (US) 1977-12-20 US disclosed
US-4060687-A Cephalosporins having a 3-α substituted alkyl grouping MERCK & CO., INC. (US) 1977-11-29 US disclosed
US-4035359-A 6α, β-Substituted penicillin derivatives MERCK & CO., INC. (US) 1977-07-12 US disclosed
US-4032521-A ANTIBIOTICS MERCK & CO., INC. (US) 1977-06-28 US disclosed
US-3974151-A Cephalosporin compounds MERCK & CO., INC. (US) 1976-08-10 US disclosed
US-3947413-A ANTIBIOTICS MERCK & CO., INC. (US) 1976-03-30 US disclosed