SCHEMBL7417451

SCHEMBL7417451

CC(C)[C@H](NC(=O)COc1cccc2ccccc12)C(=O)OCc1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 5/20 0.62
CTSD P07339 1/20 0.56
CASP1 P29466 2/20 0.54
CASP8 Q14790 2/20 0.54
CASP7 P55210 1/20 0.54
OGG1 O15527 1/20 0.52
ALDH1A1 P00352 3/20 0.52
KDM4E B2RXH2 2/20 0.52
HPGD P15428 2/20 0.52
MEN1 O00255 1/20 0.52
LMNA P02545 1/20 0.52
KMT2A Q03164 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
IL1RN P18510 1/20 0.52
ERAP2 Q6P179 1/20 0.52
ERAP1 Q9NZ08 1/20 0.52
MBTPS1 Q14703 2/20 0.51
TDP1 Q9NUW8 1/20 0.50
ADAMTS5 Q9UNA0 1/20 0.48
MAPK1 P28482 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548868 0.86 CASP3 (0.69) CASP3CTSDCASP1CASP8CASP7
SCHEMBL7419603 0.86 CASP3 (0.69) CASP3CTSDCASP1CASP8CASP7
SCHEMBL8547790 0.78 OGG1 (0.62) CASP3CASP1CASP8CASP7OGG1
SCHEMBL8547788 0.78 OGG1 (0.62) CASP3CASP1CASP8CASP7OGG1
SCHEMBL18831696 0.78 ELANE (0.41) CASP3CASP1ALDH1A1KDM4EHPGD
SCHEMBL20305851 0.78 ELANE (0.41) CASP3CTSDCASP1ALDH1A1KDM4E
SCHEMBL10208224 0.78 ELANE (0.41) CASP3CTSDCASP1ALDH1A1KDM4E
SCHEMBL8544995 0.78 CASP3 (0.60) CASP3CTSDCASP1CASP8CASP7
SCHEMBL8544998 0.78 CASP3 (0.60) CASP3CTSDCASP1CASP8CASP7
SCHEMBL6813267 0.78 CASP3 (0.57) CASP3CTSDCASP1CASP8CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993013066-A1 CYCLIC AMIDES OF 3-AMINO-2-HYDROXY-CARBOXYLIC ACIDS AS HIV-PROTEASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1993-07-08 WO disclosed