SCHEMBL7417985

SCHEMBL7417985

Cc1cc(S(C)(=O)=O)ccc1OC(F)F

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.46
PTGS2 P35354 6/20 0.44
EPAS1 Q99814 2/20 0.41
LMNA P02545 2/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
PDE4B Q07343 2/20 0.38
FAAH O00519 1/20 0.38
PTGS1 P23219 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22602047 0.80 SMN1; SMN2 (0.44) SMN1; SMN2PTGS2EPAS1ALDH1A1MAPT
SCHEMBL7412893 0.78 SMN1; SMN2 (0.67) SMN1; SMN2PTGS2LMNAALDH1A1MAPT
SCHEMBL15656580 0.78 MAPT (0.44) SMN1; SMN2PTGS2EPAS1ALDH1A1MAPT
SCHEMBL7418349 0.78 SMN1; SMN2 (0.41) SMN1; SMN2PTGS2EPAS1LMNAPDE4B
SCHEMBL29903387 0.76 SLC6A9 (0.45) SMN1; SMN2LMNA
SCHEMBL3554918 0.75 SMN1; SMN2 (0.49) SMN1; SMN2PTGS2LMNAALDH1A1MAPT
SCHEMBL7417584 0.74 PTGDR2 (0.44) SMN1; SMN2PTGS2
SCHEMBL6876872 0.74 ALDH1A1 (0.50) SMN1; SMN2LMNAALDH1A1MAPT
SCHEMBL11697683 0.73 SMN1; SMN2 (0.44) SMN1; SMN2PTGS2EPAS1LMNAALDH1A1
SCHEMBL3123667 0.73 SMN1; SMN2 (0.40) SMN1; SMN2PTGS2LMNAPDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1163214-A1 GAMMA-KETOACID DIPEPTIDES AS INHIBITORS OF CASPASE-3 Merck Frosst Canada & Co. (CA) 2001-12-19 EP disclosed
US-6225288-B1 IMPLICATED IN MODULATING APOPTOSIS; TREATMENT OF:CARDIAC AND CEREBRAL ISCHEMIA/REPERFUSION INJURY, SPINAL CORD INJURY AND ORGAN DAMAGE DURING TRANSPLANTATION, CHRONIC NEURODEGENERATIVE DISEASES, IMMUNODEFICIENCY, DIABETES, ALOPECIA, AGING MERK FROSST CANADA & CO. (CA) 2001-05-01 US disclosed
WO-2000055127-A1 GAMMA-KETOACID DIPEPTIDES AS INHIBITORS OF CASPASE-3 MERCK FROSST CANADA & CO. (CA) 2000-09-21 WO disclosed