SCHEMBL7419924

SCHEMBL7419924

CCC(=O)NCCC1COc2ccc(C(=N)N)cc21

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.54
HTR1D P28221 1/20 0.54
HTR2C P28335 1/20 0.54
MTNR1A P48039 17/20 0.47
MTNR1B P49286 17/20 0.47
ABCB11 O95342 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
USP2 O75604 1/20 0.43
NQO2 P16083 6/20 0.42
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
KLKB1 P03952 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7420409 0.83 HTR1A (0.53) HTR1AHTR1DHTR2CITGB3ITGA2B
SCHEMBL7420691 0.83 HTR1A (0.53) HTR1AHTR1DHTR2CMTNR1AMTNR1B
SCHEMBL6212650 0.83 F10 (0.51) HTR1AHTR1DHTR2CITGB3ITGA2B
SCHEMBL2640085 0.83 HTR1A (0.47) HTR1AHTR1DHTR2CITGB3ITGA2B
SCHEMBL6214226 0.82 HTR1A (0.47) HTR1AHTR1DHTR2CITGB3ITGA2B
SCHEMBL2639933 0.82 CYP1A2 (0.47) HTR1AHTR1DHTR2CITGB3ITGA2B
SCHEMBL6213779 0.82 HTR1A (0.47) HTR1AHTR1DHTR2CMTNR1AMTNR1B
SCHEMBL2639713 0.81 HTR1A (0.46) HTR1AHTR1DHTR2CMTNR1AMTNR1B
SCHEMBL6210723 0.81 HTR1A (0.46) HTR1AHTR1DHTR2CITGB3ITGA2B
SCHEMBL2640158 0.81 F10 (0.52) HTR1AHTR1DHTR2CITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222182-A2 SUBSTITUTED (AMINOIMINOMETHYL OR AMINOMETHYL) DIHYDROBENZOFURANS AND BENOZOPYRANS Aventis Pharmaceuticals Inc. (US) 2002-07-17 EP disclosed
WO-2001014358-A2 SUBSTITUTED (AMINOIMINOMETHYL OR AMINOMETHYL) DIHYDROBENZOFURANS AND BENOZOPYRANS AVENTIS PHARMACEUTICALS INC. (DE) 2001-03-01 WO disclosed