SCHEMBL7419953

SCHEMBL7419953

COc1cc2c(cc1C)CCNC2C1(c2ccco2)CC1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.46
KMT2A Q03164 5/20 0.41
MEN1 O00255 3/20 0.41
MAOA P21397 4/20 0.40
TSHR P16473 1/20 0.40
ALDH1A1 P00352 2/20 0.37
CYP2D6 P10635 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8747129 0.78 PKM (0.46) PKMKMT2AMEN1MAOATSHR
SCHEMBL7419995 0.78 MAOA (0.41) KMT2AMEN1MAOATSHRALDH1A1
SCHEMBL8549915 0.78 PKM (0.46) PKMKMT2AMEN1MAOATSHR
SCHEMBL7423986 0.77 PKM (0.45) PKMKMT2AMEN1MAOATSHR
SCHEMBL7417327 0.76 PKM (0.46) PKMKMT2AMEN1MAOATSHR
SCHEMBL8747203 0.74 PKM (0.47) PKMKMT2AMEN1MAOATSHR
Oxalic Acid SCHEMBL7418326 0.72 PKM (0.43) PKMKMT2AMEN1MAOATSHR
SCHEMBL7414016 0.69 PKM (0.46) PKMKMT2AMEN1MAOATSHR
SCHEMBL7472088 0.69 PKM (0.50) PKMKMT2AMEN1MAOATSHR
SCHEMBL7848778 0.69 MAOA (0.79) KMT2AMEN1MAOATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5807868-A ANALGESICS; PSYCHOLOGICAL DISORDES; PARKINSON*S DIESASE;COGNITION ACTIVATORS; DRUG DEPENDENCE; DYSKINESIA KNOLL AKTIENGESELLSCHAFT (DE) 1998-09-15 US disclosed
US-5804586-A ANALGESICS, PSYCHOLOGICAL DISORDERS KNOLL AKTIENGESELLSCHAFT (DE) 1998-09-08 US disclosed
EP-0707570-B1 ISOQUINOLINE DERIVATIVES AS THERAPEUTIC AGENTS KNOLL AG (DE) 1998-05-06 EP disclosed
EP-0707570-A1 ISOQUINOLINE DERIVATIVES AS THERAPEUTIC AGENTS Knoll AG (DE) 1996-04-24 EP disclosed
WO-1995000489-A1 ISOQUINOLINE DERIVATIVES AS THERAPEUTIC AGENTS KNOLL AG (DE) 1995-01-05 WO disclosed