SCHEMBL7420239

SCHEMBL7420239

COc1ccc(S(=O)(=O)N(Cc2ccccn2)S(C)(=O)=O)cc1OC

nearest known ligand 0.70

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 6/20 0.70
PDE4B Q07343 6/20 0.70
PDE4C Q08493 6/20 0.70
PDE4D Q08499 6/20 0.70
KMT2A Q03164 3/20 0.52
MEN1 O00255 2/20 0.52
MAPK1 P28482 1/20 0.52
ALDH1A1 P00352 3/20 0.49
GAA P10253 3/20 0.48
LMNA P02545 2/20 0.47
USP2 O75604 1/20 0.47
HIF1A Q16665 1/20 0.47
EPAS1 Q99814 1/20 0.47
CHRNA7 P36544 1/20 0.46
KDM4E B2RXH2 1/20 0.46
TSHR P16473 1/20 0.46
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7423813 0.88 PDE4D (0.61) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL7425474 0.84 PDE4A (0.68) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL7424509 0.82 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL7416808 0.81 PDE4D (0.73) PDE4APDE4BPDE4CPDE4DMAPK1
SCHEMBL7415074 0.77 PDE4A (0.68) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL7425188 0.77 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL7417274 0.76 PDE4A (0.55) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL7423546 0.75 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL7425459 0.75 GAA (0.80) KMT2AMEN1MAPK1ALDH1A1GAA
SCHEMBL7420807 0.74 PDE4D (0.65) PDE4APDE4BPDE4CPDE4DKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996036595-A1 3,4-DISUBSTITUTED-PHENYLSULPHONAMIDES AND THEIR THERAPEUTIC USE CHIROSCIENCE LIMITED (GB) 1996-11-21 WO claimed
EP-0986376-A1 COMPOSITIONS FOR TREATING AND PREVENTING ARTERIAL THROMBOSIS AND USE OF A FACTOR Xa INHIBITOR ON ITS OWN AND/OR COMBINED WITH A PLATELET ANTIAGGREGATING AGENT SANOFI-SYNTHELABO (FR) 2000-03-22 EP disclosed
WO-1998056365-A1 COMPOSITIONS FOR TREATING AND PREVENTING ARTERIAL THROMBOSIS AND USE OF A FACTOR Xa INHIBITOR ON ITS OWN AND/OR COMBINED WITH A PLATELET ANTIAGGREGATING AGENT SANOFI-SYNTHELABO (FR) 1998-12-17 WO disclosed
WO-1996036595-A1 3,4-DISUBSTITUTED-PHENYLSULPHONAMIDES AND THEIR THERAPEUTIC USE CHIROSCIENCE LIMITED (GB) 1996-11-21 WO disclosed