SCHEMBL7420503

SCHEMBL7420503

Cc1ccc(S(=O)(=O)N[C@@H](Cc2ccc(OCCCONC(=N)N)cc2)C(=O)OC(=O)C(F)(F)F)cc1[N+](=O)[O-]

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BCL2 P10415 8/20 0.38
ALDH1A1 P00352 2/20 0.37
MCL1 Q07820 1/20 0.37
HTT P42858 1/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
POLB P06746 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
F2 P00734 3/20 0.36
TMPRSS6 Q8IU80 3/20 0.36
MAPK1 P28482 1/20 0.35
BACE1 P56817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7414962 0.91 BCL2 (0.44) BCL2MCL1
Trifluoroacetic Acid SCHEMBL7420494 0.90 POLB (0.45) BCL2MCL1POLBITGB3ITGA2B
SCHEMBL7416087 0.89 POLB (0.37) MAPTPOLBITGB3ITGA2BF2
SCHEMBL7414953 0.88 ITGB3 (0.43) KMT2AITGB3ITGA2BF2TMPRSS6
SCHEMBL7411794 0.88 POLB (0.48) BCL2ALDH1A1MCL1POLBITGB3
SCHEMBL7418351 0.88 TYMS (0.37) MAPTITGB3ITGA2B
SCHEMBL7412096 0.87 MEN1 (0.43) ALDH1A1MEN1KMT2AITGB3ITGA2B
SCHEMBL7416574 0.87 ITGB3 (0.45) ITGB3ITGA2BF2TMPRSS6
SCHEMBL7415235 0.86 KCNA5 (0.44) SMN1; SMN2ITGB3ITGA2BF2TMPRSS6
SCHEMBL7415041 0.86 AR (0.38) BCL2MCL1MEN1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US disclosed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO disclosed