SCHEMBL7416574

SCHEMBL7416574

Cc1ccc(S(=O)(=O)N[C@@H](Cc2ccc(OCCCONC(=N)N)cc2)C(=O)OC(=O)C(F)(F)F)cc1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 6/20 0.45
ITGA2B P08514 4/20 0.45
TDP1 Q9NUW8 1/20 0.43
ITGAV P06756 2/20 0.42
ITGB1 P05556 1/20 0.42
ITGA5 P08648 1/20 0.42
F2 P00734 4/20 0.42
TMPRSS6 Q8IU80 4/20 0.42
CTSL P07711 1/20 0.40
KCNA5 P22460 1/20 0.38
HPN P05981 2/20 0.38
PLAU P00749 1/20 0.38
ST14 Q9Y5Y6 1/20 0.38
MMP2 P08253 1/20 0.37
MMP9 P14780 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7415235 0.94 KCNA5 (0.44) ITGB3ITGA2BITGAVF2TMPRSS6
SCHEMBL7694791 0.93 MMP2 (0.45) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL7699209 0.92 F2 (0.42) ITGB3ITGA2BF2TMPRSS6KCNA5
SCHEMBL7418524 0.92 F2 (0.43) ITGB3ITGA2BF2TMPRSS6KCNA5
SCHEMBL7418015 0.92 ALDH1A1 (0.46) ITGB3ITGA2BF2TMPRSS6KCNA5
SCHEMBL7413464 0.92 F2 (0.42) ITGB3ITGA2BF2TMPRSS6KCNA5
SCHEMBL7412629 0.92 CTSL (0.43) ITGB3ITGA2BF2TMPRSS6CTSL
SCHEMBL7414434 0.92 F2 (0.42) ITGB3ITGA2BF2TMPRSS6KCNA5
SCHEMBL7417592 0.91 ITGB3 (0.49) ITGB3ITGA2BITGAVF2TMPRSS6
SCHEMBL7412855 0.91 KCNA5 (0.42) ITGB3ITGA2BITGAVF2TMPRSS6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US disclosed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO disclosed