SCHEMBL7420604

SCHEMBL7420604

COC(=O)CCc1ccc2cccc(OCc3ccccc3)c2n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.51
ALDH1A1 P00352 4/20 0.50
MAPT P10636 4/20 0.50
HPGD P15428 3/20 0.50
HTT P42858 3/20 0.50
HDAC6 Q9UBN7 3/20 0.49
HDAC3 O15379 2/20 0.49
HDAC4 P56524 2/20 0.49
HDAC1 Q13547 2/20 0.49
HDAC7 Q8WUI4 2/20 0.49
HDAC2 Q92769 2/20 0.49
HDAC10 Q969S8 2/20 0.49
HDAC11 Q96DB2 2/20 0.49
HDAC8 Q9BY41 2/20 0.49
HDAC9 Q9UKV0 2/20 0.49
HDAC5 Q9UQL6 2/20 0.49
BRD4 O60885 1/20 0.48
MEN1 O00255 5/20 0.47
KMT2A Q03164 5/20 0.47
CYP1A2 P05177 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9951205 0.81 HTR1A (0.51) KDM4EALDH1A1MAPTHPGDHTT
SCHEMBL16132602 0.79 KDM4E (0.54) KDM4EALDH1A1MAPTHPGDHTT
SCHEMBL9951909 0.79 MEN1 (0.55) KDM4EALDH1A1MAPTHPGDHTT
SCHEMBL2854918 0.77 KDM4E (0.45) KDM4EALDH1A1HPGDKMT2ACYP1A2
SCHEMBL2851009 0.77 PDE10A (0.41) ALDH1A1HPGDHTTHDAC1HDAC2
SCHEMBL16106608 0.77 HDAC3 (0.49) KDM4EALDH1A1MAPTHPGDHTT
SCHEMBL16106664 0.77 HDAC3 (0.49) KDM4EALDH1A1MAPTHPGDHTT
SCHEMBL16106565 0.77 HDAC3 (0.49) KDM4EALDH1A1MAPTHPGDHTT
SCHEMBL16106558 0.77 HDAC3 (0.49) KDM4EALDH1A1MAPTHPGDHTT
SCHEMBL16106388 0.77 HDAC3 (0.49) KDM4EALDH1A1MAPTHPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999026933-A1 SUBSTITUTED AMIDINOARYL DERIVATIVES AND THEIR USE AS ANTICOAGULANTS AXYS PHARMACEUTICALS, INC. (US) 1999-06-03 WO disclosed