SCHEMBL7420635

SCHEMBL7420635

O=c1[nH]c(=O)n(-c2cccc([N+](=O)[O-])c2)c2nc(Cc3ccccc3)[nH]c12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.48
MAPT P10636 3/20 0.45
GAA P10253 2/20 0.43
RECQL P46063 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
GRIN1 Q05586 1/20 0.41
GRIN2B Q13224 1/20 0.41
PNP P00491 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
ALDH1A1 P00352 2/20 0.40
THRB P10828 1/20 0.40
PGR P06401 1/20 0.39
PDE9A O76083 1/20 0.39
PDE1C Q14123 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7604058 0.84 PNP (0.51) MAPTGAASMN1; SMN2PNPNPSR1
SCHEMBL7421927 0.84 CCNE2 (0.46) MAPTGAASMN1; SMN2PNPNPSR1
SCHEMBL7422077 0.83 PNP (0.49) MAPTGAASMN1; SMN2PNPNPSR1
SCHEMBL7421517 0.77 PNP (0.46) MAPTGAASMN1; SMN2PNPNPSR1
SCHEMBL7416425 0.74 PNP (0.47) MAPTGAASMN1; SMN2PNPNPSR1
SCHEMBL7420637 0.71 PGR (0.43) MAPTGAARECQLSMN1; SMN2PNP
SCHEMBL9432250 0.71 NPSR1 (0.49) RIPK1MAPTNPSR1MEN1KMT2A
SCHEMBL5249967 0.70 PDE4A (0.57) MAPTMEN1KMT2APDE4APDE4B
SCHEMBL10889569 0.69 PDE4A (0.57) MAPTGAAMEN1KMT2APDE4A
SCHEMBL6801649 0.69 PDE4A (0.51) MAPTGAANPSR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825993-A1 XANTHINES AND THEIR THERAPEUTIC USE Chiroscience Limited (GB) 1998-03-04 EP disclosed
WO-1996036638-A1 XANTHINES AND THEIR THERAPEUTIC USE CHIROSCIENCE LIMITED (GB) 1996-11-21 WO disclosed