SCHEMBL742178

SCHEMBL742178

COCCCn1c([C@@H]2CCCN(C(=O)[C@H]3CNC[C@H]3N(CC3c4ccccc4-c4ccccc43)C(=O)O)C2)nc2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 9/20 0.44
HRH1 P35367 8/20 0.44
CYP2D6 P10635 5/20 0.44
CHRM1 P11229 4/20 0.43
REN P00797 4/20 0.39
USP2 O75604 1/20 0.38
POLB P06746 1/20 0.38
BRD4 O60885 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL742177 1.00 KCNH2 (0.44) KCNH2HRH1CYP2D6CHRM1REN
SCHEMBL762453 0.83 HRH1 (0.39) KCNH2HRH1CYP2D6CHRM1REN
Ammonia Solution, Strong SCHEMBL741029 0.83 HRH1 (0.39) KCNH2HRH1CYP2D6CHRM1REN
SCHEMBL742179 0.81 HRH1 (0.44) KCNH2HRH1CYP2D6CHRM1USP2
SCHEMBL741382 0.80 KCNH2 (0.44) KCNH2HRH1CYP2D6CHRM1USP2
SCHEMBL741030 0.79 HRH1 (0.38) KCNH2HRH1CYP2D6CHRM1REN
SCHEMBL739857 0.78 HRH1 (0.57) KCNH2HRH1CYP2D6CHRM1USP2
SCHEMBL763016 0.75 MMP7 (0.41) KCNH2HRH1CYP2D6CHRM1
SCHEMBL738833 0.75 HRH1 (0.49) KCNH2HRH1CYP2D6CHRM1USP2
SCHEMBL738834 0.75 HRH1 (0.49) KCNH2HRH1CYP2D6CHRM1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed