SCHEMBL7422185

SCHEMBL7422185

C[C@@H]1C[N]c2ccccc2C1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.38
CREBBP Q92793 1/20 0.38
CYP2D6 P10635 1/20 0.36
MEN1 O00255 1/20 0.36
RECQL P46063 1/20 0.36
KMT2A Q03164 1/20 0.36
NOS3 P29474 2/20 0.35
NOS2 P35228 2/20 0.35
NOS1 P29475 1/20 0.35
ACHE P22303 1/20 0.34
ADRA2A P08913 2/20 0.33
ADRA2B P18089 2/20 0.33
ADRA2C P18825 2/20 0.33
CYP19A1 P11511 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
NISCH Q9Y2I1 1/20 0.32
CTSD P07339 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7422184 1.00 BRD4 (0.38) BRD4CREBBPCYP2D6MEN1RECQL
SCHEMBL5540169 0.75 CYP2D6 (0.36) CYP2D6MEN1RECQLKMT2ANOS3
SCHEMBL10388552 0.75 CYP2D6 (0.36) CYP2D6MEN1RECQLKMT2ANOS3
SCHEMBL1451031 0.75 CYP2D6 (0.43) CYP2D6MEN1RECQLKMT2ANOS3
SCHEMBL21065477 0.72 TRPA1 (0.36) BRD4CREBBPCYP2D6MEN1RECQL
SCHEMBL315647 0.71 BRD4 (0.54) BRD4CREBBPNOS3NOS2ACHE
SCHEMBL840754 0.71 NOS3 (0.47) BRD4CREBBPCYP2D6MEN1RECQL
SCHEMBL13620740 0.67 TRPA1 (0.38) BRD4CREBBPCYP2D6MEN1RECQL
SCHEMBL30358244 0.67 TRPA1 (0.38) BRD4CREBBPCYP2D6MEN1RECQL
SCHEMBL20404734 0.67 TRPA1 (0.38) BRD4CREBBPCYP2D6MEN1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0815103-A1 TRYPSIN AND THROMBIN INHIBITORS Novartis AG (CH) 1998-01-07 EP disclosed
WO-1996029327-A1 TRYPSIN AND THROMBIN INHIBITORS NOVARTIS AG (CH) 1996-09-26 WO disclosed