SCHEMBL7422369

SCHEMBL7422369

NC(=O)C1/C=C\C=C/c2ccccc2O1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.38
HPGD P15428 2/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
SIRT1 Q96EB6 4/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 2/20 0.32
LMNA P02545 2/20 0.32
MAPK1 P28482 1/20 0.32
SCN4A P35499 1/20 0.32
SCN5A Q14524 1/20 0.32
SCN9A Q15858 1/20 0.32
SIRT3 Q9NTG7 1/20 0.31
SIRT2 Q8IXJ6 2/20 0.30
MEN1 O00255 1/20 0.30
MAPT P10636 1/20 0.30
KMT2A Q03164 1/20 0.30
TRPA1 O75762 1/20 0.30
ALOX5 P09917 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7422383 1.00 ATM (0.38) ATMHPGDKDM4EALDH1A1SIRT1
SCHEMBL2971408 0.88 ATM (0.41) ATMHPGDKDM4EALDH1A1SIRT1
SCHEMBL29696802 0.88 ATM (0.41) ATMHPGDKDM4EALDH1A1SIRT1
SCHEMBL4410965 0.88 ATM (0.41) ATMHPGDKDM4EALDH1A1SIRT1
Hydrochloric Acid SCHEMBL19744196 0.87 ATM (0.40) ATMHPGDKDM4EALDH1A1SIRT1
SCHEMBL9319851 0.87 HPGD (0.37) HPGDKDM4EALDH1A1CYP2C9TSHR
SCHEMBL9319861 0.87 HPGD (0.37) HPGDKDM4EALDH1A1CYP2C9TSHR
SCHEMBL11551373 0.77 KDM4E (0.30) HPGDKDM4EALDH1A1
SCHEMBL11556600 0.74 MAOA (0.32) HPGDKDM4EALDH1A1MEN1MAPT
SCHEMBL28806661 0.74 KDM4E (0.40) ATMHPGDKDM4EALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5288731-A Antiemetics, antiserotonine agents RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1994-02-22 US disclosed
WO-1992009284-A1 2,6-METHANO-2H-1-BENZOXOCINCARBOXAMIDES AS 5-HT3-ANTAGONISTS RHONE-POULENC RORER INTERNATIONAL (HOLDINGS), INC. (US) 1992-06-11 WO disclosed