SCHEMBL7422809

SCHEMBL7422809

CN(C)c1ccc(CNC(=O)c2cc3ccccc3[nH]2)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 3/20 0.62
HDAC3 O15379 1/20 0.62
HDAC1 Q13547 1/20 0.62
NCOR2 Q9Y618 1/20 0.62
HTR2C P28335 1/20 0.62
CNR1 P21554 2/20 0.57
DRD2 P14416 1/20 0.56
DRD3 P35462 1/20 0.56
KDM4E B2RXH2 4/20 0.56
ACKR3 P25106 1/20 0.56
CA12 O43570 1/20 0.55
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
CA9 Q16790 1/20 0.55
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
ALDH1A1 P00352 2/20 0.55
GAA P10253 1/20 0.55
MAPK1 P28482 1/20 0.55
HSD17B10 Q99714 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2735969 0.85 CA12 (0.72) HDAC2HDAC3HDAC1NCOR2DRD2
SCHEMBL6657027 0.84 HDAC2 (0.67) HDAC2HDAC3HDAC1NCOR2HTR2C
SCHEMBL6657894 0.83 NHERF1 (0.69) HDAC2HDAC3HDAC1NCOR2DRD2
SCHEMBL6655159 0.83 LMNA (0.63) HDAC2HDAC3HDAC1NCOR2HTR2C
SCHEMBL25003661 0.83 KDM4E (0.57) HDAC2HDAC3HDAC1NCOR2HTR2C
SCHEMBL6656151 0.82 HDAC2 (0.62) HDAC2HDAC3HDAC1NCOR2HTR2C
SCHEMBL13587037 0.81 HDAC2 (0.67) HDAC2HDAC3HDAC1NCOR2HTR2C
SCHEMBL12584537 0.81 NAMPT (0.72) HDAC2HDAC3HDAC1NCOR2HTR2C
SCHEMBL4930492 0.81 HDAC2 (0.70) HDAC2HDAC3HDAC1NCOR2KDM4E
SCHEMBL18641772 0.81 HDAC2 (0.60) HDAC2HDAC3HDAC1NCOR2HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042287-A1 INDOLE DERIVATIVES AS INHIBITORS OF FACTOR XA Aventis Pharma Deutschland GmbH (DE) 2000-10-11 EP disclosed
WO-1999033800-A1 INDOLE DERIVATIVES AS INHIBITORS OR FACTOR XA AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 1999-07-08 WO disclosed