SCHEMBL7423496

SCHEMBL7423496

CC(C)(C)OC(=O)NC(C(=O)O)c1ccccc1O

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSS P25774 6/20 0.50
CTSK P43235 5/20 0.50
PPARA Q07869 5/20 0.44
PPARG P37231 4/20 0.44
ATM Q13315 1/20 0.44
ACE P12821 1/20 0.43
PPARD Q03181 2/20 0.43
CTSL P07711 1/20 0.42
CTSB P07858 1/20 0.42
IDO1 P14902 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15232697 0.87 CTSS (0.46) CTSSCTSKPPARAPPARGATM
SCHEMBL28505550 0.87 CTSS (0.46) CTSSCTSKPPARAPPARGATM
SCHEMBL25238924 0.85 CTSS (0.50) CTSSCTSKPPARAPPARGATM
SCHEMBL15270465 0.85 CTSS (0.50) CTSSCTSKPPARAPPARGATM
SCHEMBL27159106 0.85 CTSS (0.50) CTSSCTSKPPARAPPARGATM
SCHEMBL25282758 0.84 CTSS (0.49) CTSSCTSKPPARAPPARGATM
SCHEMBL23886560 0.84 CTSS (0.49) CTSSCTSKPPARAPPARGATM
SCHEMBL21777294 0.84 CTSS (0.49) CTSSCTSKPPARAPPARGATM
SCHEMBL265969 0.84 CTSS (0.49) CTSSCTSKPPARAPPARGATM
SCHEMBL23886587 0.84 CTSS (0.49) CTSSCTSKPPARAPPARGATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12582644-B2 O-GlcNAc transferase inhibitors and uses thereof PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2026-03-24 US disclosed
US-20210346367-A1 O-GLCNAC TRANSFERASE INHIBITORS AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2021-11-11 US disclosed
US-20210346367-A1 O-GLCNAC TRANSFERASE INHIBITORS AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2021-11-11 US disclosed
WO-2020047251-A1 O-GLCNAC TRANSFERASE INHIBITORS AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2020-03-05 WO disclosed
WO-2020047251-A1 O-GLCNAC TRANSFERASE INHIBITORS AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2020-03-05 WO disclosed
US-6225311-B1 Acetylenic α-amino acid-based sulfonamide hydroxamic acid tace inhibitors AMERICAN CYANAMID COMPANY 2001-05-01 US disclosed
US-4108854-A Process for preparing substituted glycines SMITHKLINE CORPORATION (US) 1978-08-22 US disclosed
US-3997584-A Substituted glycines and intermediates thereof SMITHKLINE CORPORATION (US) 1976-12-14 US disclosed
US-3994954-A Process for preparing substituted glycines SMITHKLINE CORPORATION (US) 1976-11-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12582644-B2 O-GlcNAc transferase inhibitors and uses thereof OGA, OGT, OSTC CTSS 1495/4885CTSK 3504/4885PPARA 4249/4885
US-20210346367-A1 O-GLCNAC TRANSFERASE INHIBITORS AND USES THEREOF OGT, OGA, UGGT1 CTSS 897/4885CTSK 1546/4885PPARA 4232/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.